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1-[4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
1-cyclopentanecarbonyl-N-(3-phenoxypropyl)piperidine-4-carboxamide
2-(oxolan-2-ylmethyl)-4-{4-[(3-phenoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(pyridin-3-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
4-(2H-1,3-benzodioxole-5-carbonyl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
6-fluoro-8-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]quinoline
1-[(2-aminopyridin-3-yl)methyl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
1-[2-(3-chlorophenyl)ethyl]-4-[(furan-3-ylmethyl)amino]pyrrolidin-2-one
1,4,6-trimethyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
3-acetamido-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]butanamide
(2R,3S,6R)-5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(dimethylamino)ethyl]-4-(hydroxymethyl)-N-[(2-methylphenyl)methyl]benzamide
3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
3-[3-(ethoxycarbonyl)-3-[(3-methoxyphenyl)methyl]piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-(3-methylthiophene-2-carbonyl)piperidine
1-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
1-[(5-chlorothiophen-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[2-(adamantan-1-yl)ethyl]-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
8-cyclopentanecarbonyl-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N,2-dimethyl-4-phenyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
(4aS,7aR)-1-[(4-ethylphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-propoxypiperidine
N,N,1-trimethyl-3-[(E)-2-phenylethenyl]-1H-1,2,4-triazol-5-amine
4-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutanamide
methyl[(5-methyl-1,2-oxazol-3-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine
(1S,5R)-6-(2-methoxyethyl)-3-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-ethyl-1-(3-methoxypropyl)-1H-1,3-benzodiazole-7-carboxamide
2-(2-methoxyethyl)-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}morpholine
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(1R,5R)-N-(3-methoxyphenyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(pyridine-3-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(4-fluoro-3-methylphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4aR,8aR)-7-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
2-(2-methyl-4-phenylpyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl]cyclopropanecarboxamide
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-({1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2,2-dimethylpropanamide
3-{[1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidin-3-yl]methyl}benzoic acid
1-(3-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
(3S,7S)-5-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
methyl 3-(4-fluorobenzamido)-6-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-cyclopropyl-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-1H-pyrrole-2-carboxamide