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2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}acetamide
2-{4-[4-(hydroxymethyl)phenyl]-1H-pyrazol-1-yl}-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-[3-methyl-4-(morpholin-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
2-(3-hydroxypropyl)-9-{imidazo[1,2-a]pyridin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{[1-(cyclohexylmethyl)-3-(dimethylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl](methyl)amino}acetate
[(1-cyclopentylpiperidin-4-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
2-{5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]but-3-enamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-5-(pyrrolidine-1-sulfonyl)benzoic acid
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N3-butyl-1-cyclohexyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
methyl (2R)-2-{[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}propanoate
1-(4-{[2-(1H-imidazol-2-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)-3-methyl-1λ6-thiolane-1,1-dione
1-benzyl-3-methyl-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-dioxa-8-azaspiro[4.5]decane
2-(pyridin-3-yloxy)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
2-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]-1,3-thiazole-4-carboxamide
1-(methoxymethyl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-azaspiro[5.5]undecan-9-amine
1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}acetamide
{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-4-yl)methanol
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
4-{4-[3-(thiomorpholin-4-ylmethyl)phenoxy]butyl}morpholine
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-(2,3-dimethylphenoxy)ethan-1-one
N-ethyl-2-[4-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperazin-1-yl]acetamide
N-(furan-2-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
methyl 3-[(4-methylphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2-methoxyphenyl)methyl]-4-(morpholin-4-yl)-N-(prop-2-en-1-yl)pentanamide
2-methyl-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepan-5-one
2-amino-1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
methyl 2-(azocane-1-sulfonyl)-6-(2,2,3,3-tetramethylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(6-methylpyridazin-3-yl)benzamide
1-{[2-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
N-[1-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-methyl-3-{methyl[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}propanamide
N-[3-(3,5-dimethylphenoxy)propyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
2-(1H-imidazol-2-yl)-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
N-[(2-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-phenyl-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4aR,8aS)-6-cyclopropanecarbonyl-decahydro-1,6-naphthyridin-1-yl]-2-(4-phenylphenyl)ethan-1-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-ethyl-3-({1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one