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N-{[4-(dimethylsulfamoyl)phenyl]methyl}-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
ethyl 2-[1-(1H-pyrrole-3-carbonyl)piperidin-2-yl]acetate
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
3-methyl-8-{2-[(2-methylphenyl)sulfanyl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1H-1,3-benzodiazol-2-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
1-cyclohexyl-4-{3-[(4-methylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-(furan-2-ylmethyl)-1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-ethylpiperazin-1-yl)-3-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
4-[2-({4-[1-(cyclohex-3-ene-1-carbonyl)piperidin-3-yl]-5-methylpyrimidin-2-yl}sulfanyl)ethyl]morpholine
3-[2-(4-fluorophenyl)ethyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
5-ethyl-2-methyl-4-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-1-yl)pyrimidine
N-[1-(2-chlorophenyl)ethyl]-3-(N-methylmethanesulfonamido)propanamide
2-(3-methylbutyl)-8-[2-(morpholin-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-1'-[(4-fluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
N-[1-(4-hydroxyphenyl)ethyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-2-(pyridin-4-yl)acetamide
2-[(3S,4R)-3-cyclopropyl-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-1-yl]acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-imidazole-5-carboxamide
3,5,7-trimethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-indole-2-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]morpholine-2-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-[(propan-2-yl)amino]pyrrolidin-2-one
{4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]morpholin-2-yl}methanamine
8-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]acetamide
5-methanesulfonyl-2-methyl-4-(piperidin-3-yl)pyrimidine
3-(4-hydroxyphenyl)-2-phenyl-N-{[(propan-2-yl)carbamoyl]methyl}propanamide
2-(4-methyl-1H-pyrazol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]benzamide
3-(2-chlorophenyl)-1-(pyridin-4-ylmethyl)-6-(1,2,5-thiadiazole-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-methoxy-3-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-2-ol
2-(5-methyl-1,3-oxazole-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-chloro-2-methylbenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
8-(1-ethyl-3-methylpiperidine-3-carbonyl)-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(cyclopropylmethyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine-3-carboxylic acid
1-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)piperidine
(2S,4R)-1-benzyl-4-{[(2,5-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-{1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[(3S,4R)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-[2-(3-methoxyphenyl)-1-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
3-hydroxy-3-({methyl[(2-methylphenyl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
2-(4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N-cyclopropyl-5-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-({[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]carbamoyl}amino)-N-(1,3-thiazol-2-yl)propanamide
(3aR,6aS)-5-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({[4-methoxy-3-(methoxymethyl)phenyl]methyl}(pyridin-2-ylmethyl)amino)butan-1-ol
{3-[3-(4-fluorophenoxy)azetidin-1-yl]-2,2-dimethylpropyl}dimethylamine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine