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9-(2,5-dimethylfuran-3-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
{4-[4-(1H-pyrazol-5-yl)phenyl]pyridin-2-yl}methanol
2-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(azocan-1-yl)-N-(2-hydroxy-3-phenylpropyl)propanamide
1-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-4-(hydroxymethyl)piperidin-4-ol
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
8-(5-acetylthiophene-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
N-[(2-fluorophenyl)methyl]-3-{1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidin-3-yl}propanamide
2-(pyridin-3-yl)-N-[(trimethylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydroquinazolin-5-amine
N-methyl-2-(3-oxo-1-{2-[4-(propan-2-yl)phenyl]acetyl}piperazin-2-yl)acetamide
methyl 3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxylate
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
methyl 4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)benzoate
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
N-cyclopropyl-3-{5-[2-(oxolan-3-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(2-aminoethyl)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-(trifluoromethyl)pyridine-3-carboxamide
2-(2-hydroxyethyl)-8-{2-[methyl(phenyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(2,3-dihydro-1-benzofuran-7-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)[(5-phenyl-1H-pyrazol-4-yl)methyl]amine
6,8-dimethyl-3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]-1,2-dihydroquinolin-2-one
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
1-methyl-2-{1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(thiophene-3-carbonyl)pyrrolidine-2-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
6-{[4-(2-methylphenyl)phenyl]methyl}-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
(4aS,8aR)-6-[1-(methoxymethyl)cyclobutanecarbonyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-benzyl-3-(2-methoxyethyl)-8-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
3-cyclopropyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-(1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)ethan-1-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
3-fluoro-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
N-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-azabicyclo[2.2.2]octan-3-amine
5-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-chloro-4-fluorophenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-(5-benzyl-2-oxo-4-propanoylpiperazin-1-yl)benzonitrile
N-(2-{[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]formamido}ethyl)acetamide
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one