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3-(4-benzylpiperazine-1-carbonyl)-N,N-dimethyl-6-(2-methylphenyl)pyridin-2-amine
N-methyl-5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)furan-2-carboxamide
1-[(4,5-dimethylfuran-2-yl)methyl]-4-(2-phenoxyethyl)piperazine
[1-(2,6,8-trimethylquinoline-4-carbonyl)azepan-2-yl]methanol
{3-[(3-chlorophenyl)methyl]-1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)piperidin-3-yl}methanol
3-benzoyl-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1H-pyrazole-3-carboxamide
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
N-(cyclobutylmethyl)-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(dimethylamino)acetamide
2-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)quinolin-8-ol
N-ethyl-4-{[(oxolan-3-yl)carbamoyl]amino}-N-phenylbenzamide
4-(4-methyl-1H-pyrazol-3-yl)-1-[(3R,5S)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperidine
1-{4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
3-methyl-1-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]butan-1-ol
4-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-2,6-dimethylphenol
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methylfuran-2-carboxamide
4-cyclopentyl-N-[2-fluoro-3-(trifluoromethyl)phenyl]-3-oxopiperazine-1-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
(2S)-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-cyclopentyl-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxopiperidine-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
(2,4,6-trimethyl-3-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}phenyl)methanol
N-ethyl-5-[4-(3-methylphenoxy)piperidine-1-carbonyl]pyrimidin-2-amine
2-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol
2-(3-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxymethyl)pyridine
2-(3-benzoylpiperidin-1-yl)-5-fluoropyridine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
4-(1H-imidazol-1-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
2-{4-[(4-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-4-[3-(oxan-4-yl)-1-propyl-1H-1,2,4-triazol-5-yl]pyridin-2-amine
5-(piperidin-4-yl)-3-[2-(propan-2-ylsulfanyl)ethyl]-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,3-diphenylpiperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(methylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
8-(5-acetyl-4-methylpyrimidin-2-yl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[2-(diethylamino)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3-{2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
7-chloro-3,5-dimethyl-N-{[4-(morpholin-4-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
(2-chlorophenyl)methyl 3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxylate
5-hydroxy-N-[4-(1H-pyrazol-1-yl)butan-2-yl]pyrazine-2-carboxamide
ethyl 4-{5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine-1-carboxylate
{9-benzyl-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
6-chloro-N-[2-(dimethylsulfamoyl)ethyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
8-(2-amino-3-fluoropropanoyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(1H-imidazol-2-ylmethyl)-5-methyl-5-phenylpiperidin-2-one
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
ethyl 5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-2-(1,3-thiazol-4-yl)acetamide
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine