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4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
2-ethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidine-5-carboxamide
(3aS,6aS)-2-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl](methyl)amino}-N-methylpropanamide
6-[3-(3-methoxyphenoxy)azetidin-1-yl]pyrimidin-4-amine
N-[(4-methoxypyridin-2-yl)methyl]-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
6-methyl-2-(4-methylphenoxymethyl)-N-(2-methylpropyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 4-[(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]benzoate
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-2-(piperidin-1-yl)acetamide
2-(dimethylamino)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(3-methylphenyl)acetamide
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}cyclopropanamine
4-[5-(5-ethoxyfuran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
ethyl 4-[(4-chlorophenyl)methyl]-1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxylate
5-chloro-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-2-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
4-phenyl-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine
4-(hydroxymethyl)-1-[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]azepan-4-ol
dimethyl({5-[3-(pyridin-4-yl)azetidine-1-carbonyl]furan-2-yl}methyl)amine
1-[4-({4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
4-[(1-butanoylpiperidin-4-yl)oxy]-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-3-methoxybenzoic acid
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-(1-benzylpiperidin-4-yl)-N-(prop-2-en-1-yl)piperidine-3-carboxamide
3-(4-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
N-(2,3-dihydro-1H-inden-1-yl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-4-methyl-2-phenylpyrimidine
1-(2-methoxyphenyl)-2,2-dimethyl-4-(oxane-4-carbonyl)piperazine
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
(3R,4R)-3,4-dimethyl-1-{2-[(4-methylphenyl)methyl]benzoyl}pyrrolidin-3-ol
4-chloro-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[5-(2-methylpropyl)-4-phenyl-1H-imidazol-1-yl]ethan-1-amine
4-[2-(1H-indol-3-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
1-(4-aminopyrimidin-2-yl)-4-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-6-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}piperidin-3-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[2-(2-chlorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4,5-dimethyl-2-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
5-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
N-methyl-5-propyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
3-{5-[(2-methoxy-5-methylphenyl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
2-(dimethylamino)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(4-methylphenyl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-[3-(thiophen-2-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(2-methylbutan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-(3-fluorophenyl)-5-[1-(1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-methyl-4-{[2-(oxan-2-yl)ethyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide