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N-[(1R,2R)-2-(benzyloxy)cyclopentyl]imidazo[1,2-a]pyridine-6-carboxamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
2-methyl-6-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydropyridazin-3-one
N-(1-{1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-({5-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-4-ol
2-(dimethylamino)-2-(2-methylphenyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
5-(cyclohex-1-en-1-yl)-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
2-[2-(aminomethyl)morpholin-4-yl]-N,N,5-trimethylpyrimidin-4-amine
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N,N,8-trimethyl-2-(1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-pyrazol-4-yl)quinoline-4-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}benzamide
(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-N,N-dimethylpyrrolidin-3-amine
2-(3-methylphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-{1-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
[(1-benzylpiperidin-4-yl)methyl]({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})propylamine
2-[1-(3-methylbutyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
5-(1-ethyl-1H-imidazol-2-yl)-1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-phenyl-1H-imidazole
1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[2-(methylsulfanyl)ethyl]piperazine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
6,7-dimethoxy-2-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-5-carboxamide
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(3-chlorophenyl)methyl]amino}pyrrolidine-2-carboxamide
methyl (2S,4R)-4-(1,3-thiazole-5-amido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
8-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-1,3-benzothiazole
2-amino-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
(2S,4R)-4-amino-1-(but-3-enoyl)-N,N-diethylpyrrolidine-2-carboxamide
N-(2-methoxy-5-methylphenyl)-2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
5-{[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]methyl}-N-methylfuran-2-carboxamide
5-{[(2,3-dihydro-1H-inden-2-yl)carbamoyl]amino}-2-methoxy-N,N-dimethylbenzamide
N-cyclohexyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
4-{3-[3-(pyridin-2-yl)azetidine-1-carbonyl]phenyl}phenol
N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
3-(azocan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
1-[2-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
1-(4-fluorophenyl)-3-methyl-5-(oxan-4-ylmethyl)-1H-1,2,4-triazole
2-cyclopentyl-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide