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8-(dimethyl-1,3-oxazole-4-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
6-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-yl)pyrimidin-4-ol
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})(3,3,3-trifluoro-2-methylpropyl)amine
methyl 2-[(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]-4-(methylsulfanyl)butanoate
1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
(2S,4R)-4-amino-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-N-methylpyrrolidine-2-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(furan-3-ylmethyl)methylamine
N-cyclopropyl-3-{[1-(4-hydroxy-4-methylpentan-2-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
(4aS,7aR)-1-(2-butoxyacetyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{5-[(2S)-2,3-dihydroxypropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-[1-(2-methylbenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
N-(3-cyano-4-ethoxyphenyl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-(2-cyclopropylpyrimidin-5-yl)-N-ethyl-N,7,8-trimethylquinoline-4-carboxamide
methyl 3-benzamido-5-[(cyclohexylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[1-tert-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]-N-methylpyrimidin-2-amine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
6-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2,4-dimethylpyridine-3-carbonitrile
3-(4-{5-[(5-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)prop-2-yn-1-ol
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-3-(methylsulfanyl)propanamide
4-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylcyclopropane-1-carboxamide
2-(3-hydroxyphenyl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclohexyl-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
2-[(2S)-2,3-dihydroxypropyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-4-carbonitrile
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
4-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1,2,3,4-tetrahydroquinolin-2-one
2-methyl-6-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
8-(2-methylpyrimidine-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
{1-[(3-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
1-(4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)-1H-imidazole
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl][1-(4-methylpyridin-2-yl)propan-2-yl]amine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-(2,3-dimethylquinoxalin-6-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
(3S,4R)-1-[(dimethylcarbamoyl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
2-(1,1-diphenylethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(3-fluorophenyl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(2-methoxyethyl)-8-[4-(thiophen-2-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[4-({1-ethyl-3-[(3-methoxyphenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
3-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
2-methyl-N-[1-(2-propoxyphenyl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(1-methylpiperidin-4-yl)ethyl]amine
(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-hydroxyacetyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-4-(trifluoromethyl)benzamide
4-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}phenol