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[2-(3,4-dimethoxyphenyl)ethyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
3-(4-hydroxyphenyl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(2S,4S)-4-amino-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-amino-3-ethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
ethyl 5-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentanoate
2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]pyridine-3-carboxamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-(4-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
1-(pyrrolidine-1-carbonyl)-4-{thieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
1-(dimethylamino)-2-{4-[(2,4,5-trimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
3-(2-chlorophenyl)-6-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
5-acetyl-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
ethyl 1-(2-methylpyridine-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
8-(1,4-dithiepan-6-yl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
1-[2-(benzyloxy)acetyl]-N,N-dimethylpyrrolidine-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
1-(3-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}phenyl)ethan-1-one
methyl[(1-{[1-(2-methylpentyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(3-methoxyphenoxy)azetidine
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[(2S,4S)-4-fluoro-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidin-2-yl]methyl}-2-methoxyacetamide
2-{4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(3-cyclopentylpropyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzoic acid
(2S,4R)-4-amino-N-methyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)thiomorpholine
1-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
ethyl 1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(quinolin-4-yl)piperidine-4-carboxylic acid
1-{4-[(1R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]piperazin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-(4-fluorophenyl)-N-[(4-methoxyphenyl)methyl]acetamide
6-amino-N-[1-(2-chlorophenyl)ethyl]pyridine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
[2,2-dimethyl-3-(morpholin-4-yl)propyl](methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
2-(phenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(5-methylfuran-2-yl)benzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)pent-4-enamide
2-(carbamoylamino)-N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]acetamide
1-benzyl-4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-6-ol
3-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]azetidin-3-yl}pyridine
2-(2-hydroxyethyl)-9-(3-methoxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide