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2-(2-{1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5-{4-[5-(oxan-2-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
3-[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]-5-fluorobenzonitrile
3-(azepane-1-carbonyl)-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-1,4-dihydropyridin-4-one
3-(2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(piperidin-3-yl)benzamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(2-methoxy-5-methylphenyl)acetic acid
5-{4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-(3-cyclopropyl-5-{pyrazolo[1,5-a]pyridin-3-yl}-1H-1,2,4-triazol-1-yl)pyridine
2-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
(1S,5R)-6-(5-fluoro-2-methoxybenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-(azepane-1-carbonyl)phenyl]-1-[1-(4-fluorophenyl)ethyl]urea
1-ethyl-4-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperazine
3-[(2-methylpyrrolidin-1-yl)methyl]-N-(quinolin-6-yl)benzamide
(1S,5S)-3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
3-hydroxy-1-(2-phenylethyl)-3-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)piperidin-2-one
N-cyclopentyl-1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)acetamide
methyl 5-[(4-hydroxybutan-2-yl)amino]-1-methyl-3-(2-phenoxyacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-1-yl}-N,N-dimethylacetamide
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-butoxy-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(azocan-1-yl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-cyclopentanecarbonyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[3-({[(2,4-difluorophenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-phenyl-1-(2,4,5-trifluorobenzoyl)piperidin-3-amine
3-{[1-(4-sulfamoylbutanoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-{[(2S,4S)-4-fluoro-1-(2-methylfuran-3-carbonyl)pyrrolidin-2-yl]methyl}-2-methylbenzene-1-sulfonamide
4-(4,6-dimethylpyrimidin-2-yl)-N-(8-methylquinolin-5-yl)piperazine-1-carboxamide
N-[3-(methylsulfanyl)propyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(3S,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-cyclopropyl-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
N4-(1H-imidazol-2-ylmethyl)-N4-methyl-6-(pyrrolidin-1-yl)pyrimidine-2,4-diamine
8-methoxy-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,5S)-5-[(pyridin-3-ylmethyl)carbamoyl]-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine-3-carboxylic acid
3-benzyl-7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
benzyl(methyl)[3-(1-methyl-1H-pyrazol-4-yl)propyl]amine
N-[(2-methoxyphenyl)methyl]-2,4-dimethyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
6-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)pyrimidin-4-amine
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
4-(2-methylphenoxy)-1-(oxolane-2-carbonyl)piperidine-4-carboxylic acid