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3-[2-(dimethylamino)ethyl]-8-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-4-amino-N,N-diethyl-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]pyrrolidine-2-carboxamide
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-5-methyl-1H-indole-2-carboxylic acid
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-oxo-2H-chromene-3-carboxamide
2-[1-(1,7-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(cyclopropylmethyl)-6-[(4-hydroxyphenyl)methyl]-3-(isoquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-[3-(5-methylfuran-2-yl)butyl]piperidine-4-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(3-methoxypropanoyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
3-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3R,4R)-1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[2-(2-chlorophenyl)-1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
1-(4-fluorophenyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-(4-methylphenyl)-3-[3-(oxolan-3-yl)propyl]urea
N5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-(3-chlorophenyl)-4-[1-(cyclohexylmethyl)piperidin-3-yl]piperazine
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(propyl)(pyridin-3-ylmethyl)amine
3-(2-methoxyethyl)-1-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}piperidine-3-carboxylic acid
2-{3-[(2-methoxyphenyl)methyl]-5-[(2-oxo-1,3-oxazolidin-3-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2,3,5-trimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(oxan-4-yl)piperidin-3-amine
(4aR,8aR)-2-(2,3-dihydro-1H-inden-2-yl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-N-(1,3,4-thiadiazol-2-yl)benzamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
N-(1,3-benzothiazol-2-ylmethyl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
4-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
2-{1-cyclohexyl-5-[(4-oxo-1,4-dihydroquinolin-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-(dimethylamino)-7-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-ol
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[5-(2-chlorophenyl)-2-methylfuran-3-carbonyl]-1,4-diazepan-5-one
3-benzyl-1-methyl-3-[2-(4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-2-one
3-[2-(3-methoxyphenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
3-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]sulfamoyl}-N-phenylbenzamide
3-(5-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-{4-[bis(4-fluorophenyl)methyl]piperazine-1-carbonyl}imidazolidin-2-one
1-butyl-4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
3-[(3R,4S)-1-(1H-indole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
1-(3-methoxy-4-methylphenyl)-3-[4-(oxolan-2-yl)butyl]urea
5-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methyl-5-(2-phenylphenyl)pent-3-yn-2-ol
2-{[(5-ethylpyridin-2-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol