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N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-(2-methoxy-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
[(2S,6S)-4-(1-phenylcyclopentanecarbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[4-(propan-2-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[(2-chloro-6-fluorophenyl)methyl]-6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-phenyl-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperidine-4-carbonitrile
4-(3-hydroxypyrrolidine-1-carbonyl)-N-(2,2,2-trifluoroethyl)benzene-1-sulfonamide
2-{2-amino-6-[(propan-2-yl)amino]pyrimidin-4-yl}benzoic acid
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
4-(3-methylphenoxy)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
1-{2-[3-(3-chlorobenzoyl)piperidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
N-{1-[({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
(3S,4R)-1-(4-carboxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(pyrimidin-2-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(4S,6R)-N-(2-methoxyethyl)-6-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
3-fluoro-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methoxy-N-methylbenzamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{octahydropyrrolo[1,2-a]piperazin-2-yl}-3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
(1R,7S)-6-(4-methylpiperazine-1-carbonyl)-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-2-(propan-2-yl)pyrimidine
8-[(2-methoxy-3,5-dimethylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[(4-fluorophenyl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
9-[(3,5-dimethylphenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-azaspiro[5.5]undecan-9-yl}-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
1-methyl-6-(pyridin-4-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(butan-2-yl)-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-chloro-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
3-(2-fluorophenyl)-5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
2-butyl-8-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
6-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[(2-methoxyphenyl)methyl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N,N-dimethyl-6-[2-(trifluoromethyl)morpholin-4-yl]pyrazine-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)quinoline-3-carboxamide
N-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
1-cyclopentyl-5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
(4aS,8aR)-1-(3-hydroxypropyl)-6-(6-methoxypyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
N-ethyl-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-4-yl)butanamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-ethylpyrimidine-5-carboxamide
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propanamide
1-{[1-(3-chloro-4-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
2-(1H-indol-3-yl)-1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one