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2-{5-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-benzyl-1-methyl-N-[(3-methylpyridin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}acetamide
2-(5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(pyridin-3-ylmethyl)acetamide
N-[4-(1H-pyrazol-5-yl)phenyl]-1-(quinolin-8-ylmethyl)piperidine-3-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyethyl)pyrrolidin-3-yl]quinoline-4-carboxamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-(3-hydroxypropyl)-1-[(2-methoxyphenyl)methyl]urea
(3S,4S)-1-(8-fluoroquinoline-2-carbonyl)-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
1-{1-[(4,5-dimethylfuran-2-yl)methyl]azetidin-3-yl}-2-methylpiperidine
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-S-(4-fluoro-2-methylphenyl)-2-oxoethane-1-sulfonamido
8-(2-methylbutyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-cycloheptylpiperidine
3,4-dimethoxy-N-[3-(1H-pyrazol-1-yl)phenyl]benzamide
1-benzyl-N3-cyclopropyl-4-oxo-N5-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-ethyl-N,5-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]thiophene-3-carboxamide
5-(2-oxo-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{3-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenyl}acetamide
N2,N2,6-trimethyl-N4-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-2,4-diamine
4-ethyl-3-({1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-tert-butyl-1-cyclohexyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-pyrazol-3-yl}phenol
(1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
5-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2-ethyl-4-methyl-1H-imidazole
methyl({[3-(methylsulfanyl)phenyl]methyl}){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
(1R,2R,6S,7S)-4-(5-propyl-1,2-oxazole-3-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-(carbamoylmethyl)-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]piperidine-3-carboxamide
8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-3-(1H-imidazol-4-yl)-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
4-[4-(5-chlorothiophene-2-carbonyl)piperazin-1-yl]quinazoline
7-(1,3-benzothiazol-2-yl)-4-[(2R)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-benzyl-3-[2-(methylsulfanyl)benzoyl]piperidine
5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
ethyl 2-[(3-{[2-(ethylsulfanyl)ethyl]carbamoyl}phenyl)amino]acetate
N-(3-{4-[(2,3-dihydro-1H-inden-1-yl)amino]piperidin-1-yl}phenyl)-4-fluorobenzene-1-sulfonamide
1-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-methyl-1,3-thiazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
(1H-imidazol-2-ylmethyl)(methyl)(3-phenylbutyl)amine
5-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(oxan-3-yl)ethyl]-4-[(propan-2-yl)sulfamoyl]benzamide
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[1-(1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2-amino-4-[3-(cyclopentyloxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(1-{6-[(cyclopropylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
1-(3-chloro-2-propoxyphenyl)-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea