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1-cyclobutanecarbonyl-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
3-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
2-amino-6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyrimidin-4-ol
2-methoxy-N-methyl-N-(1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
2-(2-hydroxyethyl)-6-(5-phenyl-1H-pyrazole-3-carbonyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-[1-(3-chloro-2-methylphenyl)-5-[(1S)-1-hydroxy-2-phenylethyl]-1H-1,2,4-triazol-3-yl]acetamide
7-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
1-(2-ethoxypyridine-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
1-(2-methoxyphenyl)-3-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
8-(5-hydroxypyrazine-2-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(4-methylphenyl)methyl]-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
N-(1-{4-[4-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-3-ol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carboxamide
2-ethyl-9-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(2-methoxyethyl)-3-[3-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclohexylmethyl)-5-[(1,4-dioxan-2-ylmethyl)(methyl)amino]azepan-2-one
3,3-dimethyl-1-{[5-(naphthalen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
5-(5-methyl-1H-indazol-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}benzoic acid
4-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-3-yl}-5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidine
2-(4-methyl-1H-imidazol-1-yl)-N-[1-(4-methylphenyl)-4-phenyl-1H-pyrazol-5-yl]acetamide
methyl 3-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-ethyl-N-methyl-5-{[(2-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-cyclobutyl-4-[(1E)-1-phenylprop-1-en-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]quinoline-4-carboxylic acid
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(1-methyl-1H-pyrazol-3-yl)piperidine
4-oxo-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-(3-ethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N,N-dimethyl-6-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}pyrazine-2-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidine-3-carboxylic acid
6-(3-fluoro-4-methoxyphenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-[2-(2-methoxyethoxy)acetamido]-N,N-dimethylazepane-1-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-[2-(thiophen-2-yl)ethyl]urea
4-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]piperazin-2-one
N-(2-methoxyethyl)-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(1H-imidazol-4-yl)ethyl]-4-(4-methoxyphenoxy)benzamide
2-(3-methoxypropyl)-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(pent-2-yn-1-yl)-4-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-3-carbonyl]-1,4-diazepan-6-ol
1-(2-methylphenyl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)-1,4-diazepane
9-(2-hydroxyethyl)-1-methyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
6-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
2-(4-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}piperazin-1-yl)phenol
1-[6-(3-methoxyphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane