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1-[(1S,5R)-6-[4-(propan-2-yl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}furan-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
3-(2,4-dimethoxybenzoyl)-1-[(5-methylthiophen-2-yl)methyl]piperidine
5-methanesulfonyl-2-methyl-N-[(4-phenyloxan-4-yl)methyl]pyrimidin-4-amine
3-(5-fluoro-2-methoxybenzoyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-phenoxypropan-1-one
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-methyl-1H-pyrazole-5-carboxamide
5-{1-[(2E)-3-(3,5-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-methyl-1H-indole-2-carboxamide
1-(2-ethylbenzoyl)-3-(1H-pyrazol-5-yl)piperidine
(1S,5R)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-ethyl-1'-(quinoxaline-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1,3-thiazole-4-carbonyl)piperidine
N-methyl-4-(4-methylpiperazin-1-yl)-N-(pyrazin-2-ylmethyl)benzamide
3-(4-methanesulfonylphenyl)-4-methyl-1,2-dihydroquinolin-2-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methoxy-N4-methyl-N4-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
N-[2-(oxolan-3-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]phenoxy}acetic acid
7-(1-benzothiophen-3-yl)-4-(3-methyl-1,2-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[1-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
1-cyclopropanecarbonyl-N-[1-(1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
(3R,4S)-4-cyclopropyl-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]pyrrolidin-3-amine
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-3-(1H-pyrazol-4-yl)propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(pyrrolidine-1-carbonyl)pyrazine
[(3R,4R)-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(1-methyl-4-phenyl-1H-imidazol-5-yl)-1H-indole
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
5-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)-2-methoxyphenol
1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-3-ethoxypropan-1-one
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(1-methylpiperidin-4-yl)piperidine
N-methyl-2,6-dioxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(4-fluorophenyl)-N-{2-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
4-[3-methoxy-5-(trifluoromethyl)phenyl]-6-methyl-2,3-dihydropyridazin-3-one
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
8-[(3-chlorophenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-(propane-1-sulfonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-fluoro-2-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
1,3-dimethyl-2,6-dioxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]pyrazine-2-carboxamide
2-{1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}pyridine
(1S,5R)-3-cyclobutanecarbonyl-6-[4-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane