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N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}morpholine-2-carboxamide
[(5-ethylfuran-2-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
7-(cyclobutylmethyl)-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
1-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
2-{3-oxo-9-[(2,4,5-trimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-(3-hydroxy-1,2-oxazol-5-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
methyl 3-{3-[2-(pyridin-2-yl)pyrrolidin-1-yl]propanamido}thiophene-2-carboxylate
6,7-dimethoxy-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-amine
2-methoxy-3-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrazine
3-methyl-7-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-methyl-7-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-{[1-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(prop-2-en-1-yl)-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(4-methoxy-3-methylphenyl)-1H-pyrazol-1-yl]-N-methylacetamide
(1-benzothiophen-2-ylmethyl)[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
(1S,4S)-2-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-2-azabicyclo[2.2.1]heptane
benzyl(cyclobutylmethyl){[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-(4-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}phenyl)acetamide
1-(cyclohexylmethyl)-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-2-one
6-methoxy-4-methyl-2-[2-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrrolidin-1-yl]quinazoline
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
3-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)propan-1-ol
7-(6-chloro-2-methylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-[2-(3-methoxyphenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
7-methyl-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-[1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)azetidin-3-yl]pyridine
ethyl 1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(3-phenylpyrrolidin-1-yl)ethyl]amine
N-[(3S,4R)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)-2,6-dimethoxyphenol
3-(cyclopropylmethyl)-1-[2-(morpholin-4-yl)benzoyl]piperidine-3-carboxylic acid
ethyl 2-(4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
2-amino-3-ethyl-N-[1-(3-methylphenyl)piperidin-4-yl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(1-phenylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[(3-fluorophenyl)methyl]-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]piperazin-2-one
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
7-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
N-[3-(1H-imidazol-5-yl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-2-oxopentanamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1H-indole-6-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(pyridin-3-ylmethyl)furan-3-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-2-methoxyacetamide
[(4-fluorophenyl)methyl]({[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl})methylamine