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3-(3-hydroxy-3-methylbutyl)-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]benzamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide
(1S,3R)-3-amino-N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]cyclopentane-1-carboxamide
2-methoxy-N,N-dimethyl-5-({[3-(methylsulfanyl)propyl]carbamoyl}amino)benzamide
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-N-[3-(oxolan-3-yl)propyl]piperidin-4-amine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
2-{3-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]phenoxy}acetamide
N-(4-fluorophenyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-amine
(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-methoxypiperidin-4-amine
3-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecane
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(4-fluorophenyl)piperazine
2-(phenylsulfanyl)-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(1-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}piperidin-4-yl)-2-methylpropan-1-ol
2-benzyl-8-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}but-2-yn-1-one
2-ethyl-4-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-5-carboxamide
4-(4-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
3-(4-hydroxyphenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-{4-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-1-yl}propanamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
(3S)-1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-ol
1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
2-(1-methyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
N-(2-cyclobutyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-(trifluoromethyl)benzamide
4-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1,4-oxazepan-6-ol
2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]pyrimidin-4-amine
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-(cyclobutylmethyl)-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(1-cyclopropylpropan-2-yl)piperidine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
N-cyclohexyl-2-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)quinazolin-4-amine
(2R,3S,6R)-5-benzyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-hydroxy-3-methyl-N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}benzamide
1-(3-phenyl-1H-pyrazole-5-carbonyl)-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-N-(thiophen-2-ylmethyl)propanamide
2-{[(4,6-dimethylpyrimidin-2-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
(3R,5S)-1-benzyl-N-{[4-(dimethylamino)phenyl]methyl}-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-chloro-5-acetamido-N-methyl-N-(thiophen-3-ylmethyl)benzamide
N-(3-methoxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
9-ethyl-1-methyl-4-[2-(methylsulfanyl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(2-hydroxy-4-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-{4-[(5-ethylfuran-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide