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1-cyclohexyl-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
4-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}pyrimidin-2-amine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-({7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-{1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-3-yl}propan-1-one
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopropanecarboxamide
{imidazo[1,2-a]pyridin-2-ylmethyl}[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
methyl (2R)-2-[6-(diethylcarbamoyl)-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl]propanoate
2-cyclopentyl-N-{7-[4-(methoxymethyl)piperidine-1-carbonyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazol-5-yl}acetamide
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-benzyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(5-{[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-(4-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(quinoline-2-carbonyl)piperidin-3-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-[6-(methoxymethyl)pyrimidin-4-yl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
1-benzyl-3-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-methylbutyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
4-[(1-carbamoylcyclopentyl)sulfamoyl]-N-(2-methylpropyl)benzamide
N-(4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
1-[4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
6-cyclopentyl-3-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
ethyl 1-[(3-acetylphenyl)carbamoyl]-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
methyl 6-benzyl-2-[(4-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{4-[(4-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-one
1-(4-fluorophenyl)-2,2-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}cyclopropane-1-carboxamide
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-[(4-ethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 4-(2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamido)butanoate
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(oxan-4-ylmethyl)piperidine
7-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
6-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-methyl-6-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
5-cyclopropanecarbonyl-1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(2,3-dihydro-1H-inden-2-yl)-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-[4-(4-fluorophenoxy)piperidin-1-yl]-5-(4-fluorophenyl)-1,2,4-triazine
2-(1,2,3,6-tetrahydropyridin-4-yl)-N-{[1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl}acetamide
N-(furan-3-ylmethyl)-N,5-dimethyl-2-(2-methylpropanamido)benzamide
1-({4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
3-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-1-[3,5-difluoro-4-(trifluoromethyl)phenyl]urea
7-fluoro-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[3-(methylsulfamoyl)phenyl]-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
3-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-{4-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]thiophen-2-yl}ethan-1-one
2-amino-6-(4-{[2-(furan-2-yl)phenyl]methyl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
5-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-indole
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(3-methylpyridin-2-yl)methyl]-2-phenylacetamide
2-amino-4-(3-chloro-4-hydroxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile