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N,N-dimethyl-1-[2-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-amine
8-(1-methyl-1H-imidazole-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2-chloro-6-methoxy-4-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}phenoxy)acetamide
7-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(4-{2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazin-1-yl)-N,N-dimethylacetamide
3-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-(1H-1,2,4-triazol-3-yl)urea
methyl (2S,4R)-4-[3-(4-fluorophenyl)benzamido]-1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)-2-(pyrrolidin-3-yl)acetamide
(3R,4R)-N-cyclopentyl-3-hydroxy-3,4-dimethylpyrrolidine-1-carboxamide
(1-methyl-1H-imidazol-2-yl)(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)methanol
3-{4-[(3-phenyloxolan-3-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
5-methyl-N-{2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl}pyrazine-2-carboxamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(1H-1,2,4-triazol-3-yl)benzamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-(thiophen-3-ylmethyl)propanamide
5-(3-phenylpropyl)-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-[(3-methoxyphenyl)methyl]-3-methyl-5-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
4-[4-(4-chlorobenzoyl)piperazin-1-yl]-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N,1,3-trimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(1,4-oxazepane-4-carbonyl)-2-(pyridin-4-yl)quinoline
5-fluoro-2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
(3E)-1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pent-3-en-1-one
4-(1-benzothiophen-2-ylmethyl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
1-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenylpiperidin-4-yl]ethan-1-one
3-{[1-(1-methylpiperidin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1H-indole
1-{2-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-(3-chloro-4-methoxyphenyl)-6-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 4-{[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}butanoate
2-(7,8-dimethyl-4-oxo-3,4-dihydroquinazolin-3-yl)acetic acid
1-(2-methoxyphenyl)-3-(2-methylpropyl)-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-1,2,4-triazole
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{2-chloro-4-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]phenoxy}acetamide
5-cyclopropyl-N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-1,3,4-oxadiazol-2-amine
1-cyclopropyl-4-[4-(2-methylpyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
9-(3-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
{1-[(2-fluoro-5-methoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-ethyl-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-N-(pyridin-4-ylmethyl)piperidin-3-amine
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
(2S,4S,5R)-5-(3-chlorophenyl)-4-[(1H-imidazol-2-ylmethyl)(methyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
1-(3-chloro-2-methylphenyl)-3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
2-(4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
N-methyl-N-(quinoxalin-2-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
methyl 5-[(3-methylbutyl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-(ethanesulfonyl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
N-tert-butyl-1-cyclohexyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-chloro-N-cyclopentyl-4-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(furan-2-yl)ethane-1,2-dione