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N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(2-oxopiperidin-1-yl)acetamide
N-cyclohexyl-3-(3-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-(1-{4-[2-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
5-{[(butan-2-yl)(methyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
ethyl N-[4-(3-fluoro-4-methylphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]carbamate
1-(methoxymethyl)-N-[(3R,4S)-4-propyl-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-3-yl]cyclobutane-1-carboxamide
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-(3,4,5-trifluorophenyl)piperidine-1-carboxamide
4-(7-chloroquinolin-4-yl)-2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenol
(1R,5R)-3-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
[(1R,3S,3aS,6aR)-3-(2,5-dimethoxyphenyl)-5-methyl-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{3-[(1,3-thiazol-2-ylmethyl)amino]phenyl}pyrrolidin-2-one
4-methyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-1,2,3-thiadiazole-5-carboxamide
3-methyl-3-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
1-(pyridin-3-yl)-2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethan-1-ol
2-ethoxy-6-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
6-fluoro-2-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}quinolin-4-ol
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(1H-1,2,4-triazol-3-yl)benzamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(methoxymethyl)piperidine
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyrimidin-2-amine
2-phenoxy-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(methoxymethyl)pyrimidine
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl[2-(methylsulfanyl)ethyl]{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-[3-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propyl]-6-methyl-1,2-dihydropyridin-2-one
2-[2-(4-fluorophenyl)ethyl]-4-{4-[2-(naphthalen-2-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-cyclopentyl-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
1-cyclopropanecarbonyl-3-[2-(2-fluorophenyl)ethyl]piperidine
1-[(3-hydroxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-methyl-6-[5-(2H-1,2,3,4-tetrazol-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
(4aS,7aR)-1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-{[(3-phenylpropyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
ethyl 1-methyl-5-[2-(pyridin-4-yl)quinoline-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-ethyl-3-{[1-(3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-chloro-N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}pyridine-4-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(furan-2-carbonyl)piperidine-3-carboxylate
N-{4-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)-1,2,3-thiadiazole-4-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-[2-(ethylsulfanyl)phenyl]urea
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
6-[(3,5-dimethylphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(pyridin-3-yl)-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrimidin-4-ol
3-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)pyrrolidin-3-ol
3-(4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
1-cyclobutanecarbonyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
1-(cyclohexylmethyl)-5-[(1-methylpyrrolidin-2-yl)methyl]-1H-1,2,4-triazole
[(3-methoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine