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1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-decahydroisoquinoline
1-methyl-3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
methyl 3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2,5-dioxoimidazolidin-4-yl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}propanamide
N-[(2-methoxyphenyl)methyl]-N-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}cyclopropanamine
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
5-[(dimethylamino)methyl]-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]furan-2-carboxamide
5-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
4-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-cycloheptyl-4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1,7-dimethyl-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1H-indole
1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
8-(1-benzofuran-2-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]piperazine
(3aS,6aR)-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(5-methyl-2-phenylfuran-3-carbonyl)piperidine
N-butyl-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(3R,4R)-1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
[9-(cyclopropylmethyl)-3-(2-methylpyrimidine-5-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
[(5-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(3S,4R)-1-[3-(3-chlorophenyl)propanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
5-{[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
1-methanesulfonyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
(3S,9aR)-8-(3-methoxybenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,N-dimethyl-2-(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)acetamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}acetamide
[(1-cyclopentylpiperidin-3-yl)methyl][(1-methyl-1H-1,3-benzodiazol-2-yl)methyl][2-(piperidin-1-yl)ethyl]amine
(5S)-5-{[benzyl({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-6-methylquinoline-4-carboxamide
[1-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-2-yl]methanol
9-(6-methylpyridazin-3-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-(3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-phenylpropanamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethoxyethan-1-one
1-(pyridin-2-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-(1H-pyrazole-4-carbonyl)piperidine
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
2-(2-chloro-4-fluorophenyl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}acetamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[5-(morpholin-4-yl)pentyl]propanamide
1-(1-cyclopropanecarbonylpiperidin-3-yl)-3-(2,4-dimethoxyphenyl)urea
2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide