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(3aS,7aR)-2-{[6-(dimethylamino)pyridin-3-yl]methyl}-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3R,4R)-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
8-[(3-methylpyrazin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
(2S,4S)-1-(cyclopentylmethyl)-N-ethyl-4-[2-(3-methylphenyl)acetamido]pyrrolidine-2-carboxamide
7-(2,3,6-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(dimethylamino)-N-(1-ethoxy-2-methylpropan-2-yl)-2-(3-fluorophenyl)acetamide
methyl (2S,4R)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
3-(5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
1-(cyclopropylmethyl)-5-(2,3-dihydro-1-benzofuran-2-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 1-(2-acetamidoacetyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-(3,4,5-trimethoxyphenyl)-2-azaspiro[4.4]nonane-2-carboxamide
8-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]quinoline
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
3-({1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzoic acid
1-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}-4-phenylbutane-1,4-dione
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)furan-2-carboxamide
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
4-(4-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
1-methyl-2-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,3-benzodiazole
2-[2-chloro-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propanoic acid
6-cyclopropyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methylpyrimidin-4-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-2-yl)acetamide
benzyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
N-[2-(dimethylsulfamoyl)ethyl]-3-(4-fluorophenyl)-3-phenylpropanamide
2-[2-(1H-imidazol-1-yl)ethyl]-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
(1R,5R)-3-(2-butoxybenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]azepane-2-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
ethyl 2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
3-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-indole
1-[2-({4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethyl]imidazolidin-2-one
1-(4-fluoro-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](quinolin-5-ylmethyl)amine
(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
5-chloro-2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenol
4-{7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
6-methyl-2-[({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]quinolin-4-ol
N-{2-methyl-1-[7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}pyridine-2-carboxamide
methyl 2-(5-{1-[(2-methoxypyridin-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
2-methyl-4-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenyl)butan-2-ol
4-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}phenol
6-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
1-(4-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
2-(dimethylamino)-N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)acetamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-(5-methylthiophen-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide