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methyl 3-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-benzyl{[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]amino}sulfonamide
1-[3-(2-methoxyphenyl)propanamido]cyclopentane-1-carboxylic acid
5-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]isoquinoline
2-ethyl-9-[(5-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-(4-methylbenzenesulfonamidomethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-methyl-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-(quinolin-6-ylmethyl)acetamide
(3S,4S)-1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-phenyl-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
5,7-dimethyl-4-(piperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(1S,4S)-2-benzyl-5-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2,5-diazabicyclo[2.2.1]heptane
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
9-[3-(pyridin-2-yl)propanoyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[(2,4-diethoxy-3-methylphenyl)methyl]-4-(hydroxymethyl)piperidin-3-ol
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-methoxyphenoxymethyl)piperidine
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
2-[(3,4-difluorophenyl)methyl]-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[(4-sulfamoylphenyl)methyl]acetamide
2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
5-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
3-[1-(isoquinoline-5-carbonyl)piperidin-3-yl]benzoic acid
1-ethyl-2-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole
ethyl 1-(3-phenylpropyl)-5-[3-(pyridin-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-[(1R,5R)-6-{[3-(2-hydroxyethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-(1-propyl-1H-pyrazol-5-yl)urea
N-[2-(3-methoxyphenyl)-1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
3-[(3-methyloxetan-3-yl)methyl]-1-[4-(propylsulfanyl)phenyl]urea
5-[1-(3-chlorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(5-{1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
1-(isoquinoline-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(2-hydroxyphenoxy)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
1-(2,3-dimethylbenzoyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
[3-(cyclopropylmethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl]methanol
N-(2-methoxyethyl)-N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)thian-4-amine
(3S,4R)-4-(2-methoxyphenyl)-1-(2-methoxypyridine-4-carbonyl)pyrrolidine-3-carboxylic acid
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-cyclohexylethan-1-one
(2S,4S)-4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-ol
2-(4-methoxyphenyl)-2-[4-(morpholine-4-carbonyl)piperidin-1-yl]acetic acid
methyl 5-{2,7-diazaspiro[4.5]decane-2-sulfonyl}-1-methyl-1H-pyrrole-2-carboxylate
5-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine