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N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]acetamide
4-{[3-(4-phenyl-1H-imidazol-5-yl)phenyl]methyl}morpholine
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4R)-1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-methylpiperidine-3,4-diol
(2S,4S)-N-ethyl-4-[2-(3-fluoro-4-hydroxyphenyl)acetamido]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-methyl-3-(2-methylphenyl)-3-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
3-{4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carbonyl}piperidine-1-carboxamide
1-[2-(2-methoxyphenoxy)ethyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-ethoxy-1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]propan-1-one
(4aS,7aR)-1-(1,2,4-oxadiazol-3-ylmethyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-[1-(pentan-3-yl)-1H-pyrazol-5-yl]urea
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(naphthalen-1-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methyl-1H-1,3-benzodiazole-5-carboxamide
2-[4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
1-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyrrolidin-2-one
1-[(4-fluorophenyl)methyl]-4-(5-phenyl-1,2-oxazole-4-carbonyl)-1,4-diazepane
N-{3-[4-({[3-(furan-2-yl)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}pyrazine-2-carboxamide
N-cyclopropyl-3-(2-fluorophenyl)-N-(1H-indol-5-ylmethyl)-1H-pyrazole-5-carboxamide
3-[(dimethylamino)methyl]-1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidin-3-ol
4-cyclopentyl-3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
7-(3-chlorophenyl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(4-methylpiperazin-1-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
methyl 3-[(2-ethoxyphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(1H-1,3-benzodiazol-1-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]propanamide
3-(cyclopropylmethyl)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidine-3-carboxylic acid
methyl 1-{3-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
2-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-3-carboxamide
2-[1-(3,4-difluorophenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
(5-methyl-7-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
(3S,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[4-(propan-2-yl)phenyl]methyl})(pyridin-4-ylmethyl)amine
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-fluorophenyl)ethyl]acetamide
1-{4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}ethan-1-one
4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]thiomorpholine
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazole
4-[1-(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)piperidine-3-carbonyl]morpholine
1-(pyridin-3-yl)-4-(4,4,4-trifluorobutyl)piperazine
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
8-cyclopropyl-N-[(2-methylphenyl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-6-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
8-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-(piperidin-1-yl)quinoline
1-(diethylamino)-3-(5-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)azetidin-3-ol