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4-[2-(ethylamino)pyrimidine-5-carbonyl]-3-(3-fluorophenyl)piperazin-2-one
5-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1,6-dimethyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
5-[3,5-dimethyl-4-(2-oxopropyl)-1H-pyrazol-1-yl]-N,N-diethylfuran-2-carboxamide
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}azetidin-3-ol
5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
N-(1,3-dihydroxypropan-2-yl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-methyl-2-(piperidin-1-yl)pyrimidine-5-carboxamide
4-{6-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}-1,3-dimethylpiperazin-2-one
4-methanesulfonyl-N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}piperazine-1-carboxamide
4-[5-(1-methyl-2-oxoimidazolidin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
1-methyl-N-(2-phenylethyl)-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(dimethylamino)phenyl]-3-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
N-(1-{4-[3-(1H-pyrazol-1-yl)phenyl]phenyl}ethyl)acetamide
(1S,5R)-3-[(5-fluoro-2-methoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-2-[(2-methoxyphenyl)methyl]-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
[(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
3-[5-(carbamoylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopentylpropanamide
1-cyclopentyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-chloro-4-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)benzamide
9-(oxane-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
5-(2-fluorophenyl)-3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-1,2,4-triazine
3-[(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
1-{2-hydroxy-3-[2-methoxy-4-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1-{[3-chloro-4-(2,3-dihydro-1,4-benzodioxin-6-yloxy)phenyl]methyl}pyrrolidine
(1S,4S)-2-(3-chlorophenyl)-5-(dimethyl-1,3-oxazole-5-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-cyclohexyl-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-chloro-N-[1-(pyrimidin-2-yl)piperidin-3-yl]thiophene-2-carboxamide
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}thiophene-3-sulfonamide
methyl 5-(cyclohexylamino)-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenyl)piperidine
4-({2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
N-[(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-hydroxyazepan-4-yl)methyl]methanesulfonamide
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
5-(3-methoxyphenoxymethyl)-3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrimidin-2-yl)-1,4-diazepane
1-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1,3-dimethyl-6-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-methoxy-1-{4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
[(2S,4R)-4-(dimethylamino)-1-[(1-ethyl-1H-indol-5-yl)methyl]pyrrolidin-2-yl]methanol
N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
8-[(2-aminopyridin-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide