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3-(3-fluorophenyl)-4-[3-(2-oxopiperidin-1-yl)propanoyl]piperazin-2-one
2-(3-methoxypropyl)-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
6-fluoro-2-({[(2S)-1-hydroxy-4-methylpentan-2-yl]amino}methyl)quinolin-4-ol
3-{[2-(3-fluorophenyl)ethyl]sulfamoyl}-N-(2-methoxyethyl)benzamide
2-chloro-N-{[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}benzamide
4-ethyl-3-(1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-2-phenylethan-1-ol
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-phenylethan-1-one
N-[(8-methoxyquinolin-5-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
3-butanamido-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]benzamide
3-ethyl-1-methyl-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
[1-(2-{[2-(morpholine-4-carbonyl)pyridin-4-yl]amino}ethyl)piperidin-2-yl]methanol
4-benzyl-1-(2-oxo-2H-chromene-3-carbonyl)-1,4-diazepan-5-one
5-(1,4-dioxan-2-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazole
2-(3-methoxyphenoxy)-5-(4H-1,2,4-triazol-4-yl)pyridine
3-(oxolan-3-yl)-5-(5-phenoxyfuran-2-yl)-1,2,4-oxadiazole
3-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
N-[2-(3-methoxyphenyl)-1-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]ethyl]-N-methylpyridine-2-carboxamide
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]acetamide
4-(4-methanesulfonylphenyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
methyl 2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]acetate
N-(2-{2-azabicyclo[2.2.1]hept-5-en-2-yl}ethyl)-2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carboxamide
4-methyl-2-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
N-[(4-chlorophenyl)methyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropan-1-amine
2-(cyclopentylmethyl)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
(2-{5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-3-methyl-1H-pyrazol-1-yl}ethyl)dimethylamine
9-(1-benzoylpiperidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidine-2,4-diamine
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
4-(1H-pyrazol-4-yl)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]butan-1-one
N-(1-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(2-fluorophenyl)acetamide
3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}isoquinoline
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
4-[6-(piperidin-1-yl)pyrimidin-4-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
2-methyl-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]-1,4-diazepan-5-one
4-[3-(dimethylamino)benzoyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
methyl 2-{1-[(8-hydroxyquinolin-2-yl)methyl]-3-oxopiperazin-2-yl}acetate
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidine-4-carboxylate
[(2S)-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
4-[(1-{[1-(thian-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one