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2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
5-ethyl-2,4-dimethyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-(2,3-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(2E)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenyl-N-(propan-2-yl)prop-2-enamide
3-{3,5-dimethyl-1-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrazol-4-yl}propanoic acid
2-(2-methoxyacetamido)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)benzamide
ethyl 1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
3-(4-fluorophenyl)-4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(thiophen-2-yl)propan-1-one
1-[(2-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-(hydroxymethyl)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-3-ol
3-[2-(2-hydroxyethoxy)ethyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
(5S,9aS,9bS)-5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridine-2-carbonitrile
1-[2-(4-chlorophenyl)ethyl]-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
3-tert-butyl-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(4-ethylpiperazin-1-yl)-3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]propan-1-one
(8R,9aS)-8-hydroxy-2-{[2-(trifluoromethyl)phenyl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-[2-(diethylamino)ethyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(2-{1-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-(1H-imidazol-4-ylmethyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
4-amino-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine-5-carbonitrile
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-sulfamoylbutanamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
4-[(2-cyclopropyl-1H-imidazol-1-yl)methyl]-1-(2-phenylethyl)piperidine
3-(2-ethoxyethyl)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-2,4-dimethylpyrimidine
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
(3aR,6aS)-1-oxo-2-propyl-5-[(thiophen-2-ylmethyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-benzofuran-2-carboxamide
1-{1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
4-(3-fluoro-4-hydroxy-5-methoxyphenyl)-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
N-(oxolan-3-ylmethyl)-4-(1H-1,2,3,4-tetrazol-5-yloxy)aniline
(3R,4S)-4-cyclopropyl-1-(4-fluoro-2-methylbenzenesulfonyl)pyrrolidin-3-amine
ethyl 1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
N-(3-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
N-({1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl}methyl)-3-phenylpropanamide
3-[2-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(1,3-thiazol-4-ylmethyl)amine
N-(1-cycloheptylpiperidin-3-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-5,6,7,8-tetrahydroquinoxaline
4-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
2-{2-[3-(dimethylamino)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
(3R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
5-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-benzofuran-2-carboxamide