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N-ethyl-2,4-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrimidine-5-carboxamide
[1-(3-{3H-imidazo[4,5-b]pyridin-6-yl}phenyl)ethyl]dimethylamine
N-(9H-fluoren-9-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-2,6-dimethylphenol
8-(3-fluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(pyridin-3-yl)-4-[(1H-1,2,4-triazol-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(4-chloro-3-methylphenyl)-2-({2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}amino)acetamide
2-[(2-fluorophenyl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
4-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
2-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]propanamide
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-methyl-1-{1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}propan-1-ol
3-[5-(4-cyclopentylpyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-[1-(2,4-dimethylphenyl)-1H-pyrazol-4-yl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
methyl 2-{[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-4-(methylsulfanyl)butanoate
2-cyclopropyl-9-[(6-methylpyridin-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[5-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)furan-2-yl]-1H-pyrazole
(2S,4S)-4-(3-fluorobenzamido)-1-methyl-N-(3-phenylpropyl)pyrrolidine-2-carboxamide
N-[2-(5-methyl-4-{[methyl({[4-(trifluoromethoxy)phenyl]methyl})amino]methyl}-1,3-oxazol-2-yl)phenyl]methanesulfonamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-8-methoxyquinoline
9-[(1,5-dimethyl-1H-indol-2-yl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[5-(pyridin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(but-2-ynoyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-(5-methoxy-2-{[(thiophen-3-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-methylpyrimidine-5-carboxamide
4-[(4-methoxyphenyl)methyl]-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
1-[(2-fluorophenyl)methyl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-methoxy-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
1-ethyl-N-[(5-methylfuran-2-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-ethyl-3-methylpiperazin-2-one
N-(oxolan-2-ylmethyl)-3-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}propanamide
N-[(6-methylquinolin-5-yl)methyl]-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-({[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)-3,5-dimethylpyridin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-methoxyphenyl)methyl]acetamide
N'-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}butanediamide
[(3R,4R)-1-(4-chlorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(1-cyclopentyl-4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
(3R,5S)-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-ethylbutanamide
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(pyrrolidin-3-yl)acetamide
2-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]pyridine-4-carbonitrile
5-acetyl-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-3-carboxamide
N-ethyl-N-(2-methoxyethyl)-2-propyl-1,3-thiazole-4-carboxamide
N-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}aniline