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N-(3-chloro-4-propanamidophenyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(1S,5R)-6-benzyl-3-(2-methyl-6-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-benzyl-N-(2-hydroxyethyl)propanamide
6-cyclopentyl-2-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-(1-propyl-1H-pyrazol-5-yl)benzamide
4-benzyl-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(3-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}quinoline
1-[2-(oxan-2-ylmethoxy)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3-chlorophenyl)-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
(3aR,6aS)-5-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
8-[2-(dimethylamino)benzoyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxo-N-(1,3-thiazol-2-yl)acetamide
4-methoxy-3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
5-methyl-4-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
3-chloro-N-(2-methoxyethyl)-4-{[1-(oxolan-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-acetamido-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}benzamide
1-(2-fluorophenyl)-3-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[1-(cyclohexylmethyl)-4-[1-(4-fluorophenyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N,N-diethyl-1-({4-[(3-hydroxy-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
2-[5-(3-ethynylphenyl)-1,2,4-oxadiazol-3-yl]pyrazine
1-[2-({[2-(4-chlorophenyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-hydroxypyridine-3-carboxamide
3-chloro-4-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-benzothiophene-2-carboxamide
ethyl 4-[4-(2-methylpropyl)-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl]piperidine-1-carboxylate
3-(6-phenylpyridazin-3-yl)-3,9-diazaspiro[5.5]undecane
N-(1-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-3-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
(2R)-2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}propanamide
N-(1-{2-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-fluorobenzamide
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
N1,N1-dimethyl-N3-{[1-(phenoxymethyl)cyclopropyl]methyl}piperidine-1,3-dicarboxamide
4-(4-fluorophenyl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}oxane-4-carboxamide
1-benzyl-5-{[2-(diethylamino)ethyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(4aR,7aS)-4-(1H-imidazol-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(propan-2-yl)pyrimidine-4-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
(1R,5S,8R)-3-[(2-cyclohexylpyrimidin-5-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
5-(azepane-1-carbonyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,6-difluorobenzamide
1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})amine
5-chloro-2-fluoro-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)benzamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-(2-methoxyphenyl)propanamide