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(1R,5R)-N-[(4-chlorophenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
ethyl 1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-1-(2-chlorophenyl)piperazin-2-one
1-(3-chloro-4-ethoxyphenyl)-3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)urea
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(1R,5R)-6-(2-methoxyethyl)-3-[2-methyl-5-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-phenyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-amine
8-[2-(2-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3-{4-[3-(methylamino)pyrazin-2-yl]phenyl}propanoic acid
methyl 3-(1-benzofuran-2-ylmethyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-benzyl-2-[4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1H-pyrazole-3-carboxamide
1-(1-butylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 1-benzyl-5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
5-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)isoquinoline
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 6-[(3,4-difluorophenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{4-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
3-cyclohexyl-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1H-pyrazole
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
(2E)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(thiophen-2-yl)prop-2-enamide
N-cyclopropyl-1-[1-(2-oxo-4-phenylbutanoyl)piperidin-4-yl]piperidine-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-2-yn-1-one
N-({7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
6-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-oxo-N-(thiophen-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(pyridin-2-yl)ethyl]benzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-(3-acetyl-1H-indol-1-yl)-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
2-methyl-6-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)pyrimidin-4-ol
3-(oxolan-3-yl)-5-[1-(propan-2-yl)-1H-pyrrol-2-yl]-1,2,4-oxadiazole
2-(2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
1,4-dimethyl-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-(2-chloro-4-fluorophenyl)-1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)ethan-1-one
2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
4-benzyl-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-ethyl-1,4-diazepan-5-one
ethyl 2-(4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
1-benzyl-8-[(2E)-2-methylbut-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(cyclohexylmethyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
3-(2-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)propanamide
(1S,5R)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)formamido]-3-(4-fluorophenyl)propanoic acid