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5-(ethylsulfanyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}thiophene-2-carboxamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(1,2-oxazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(cyclohexylmethyl)-5-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-azaspiro[4.4]nonane
4-({[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-(2-{8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-ol
3-{[3-(2-fluorophenyl)-3-phenylpropanamido]methyl}-1,2,4-oxadiazole-5-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}[(1-ethylpyrrolidin-3-yl)methyl]methylamine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(3-methylpentanamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepane
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H-imidazole-5-carboxamide
methyl (2S)-3-methyl-2-[3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamido]butanoate
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholine-2-carboxylic acid
5-{[(3R,4S)-3-(3-methoxypropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
methyl 4-[5-({ethyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(3S,4S)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N1-[4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pentane-1,5-diamine
4-{4-[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenol
(3R,4S)-4-cyclopropyl-1-[3-(methoxymethyl)benzoyl]-N,N-dimethylpyrrolidin-3-amine
N-(pyridin-2-ylmethyl)-3-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(2-methyl-1-{7-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxolane-3-carboxamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(methylamino)ethyl]amine
11-{[(3-fluorophenyl)methyl]amino}-4-[2-(3-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-methyl-3-[3-(3,4,5-trimethoxyphenyl)phenyl]-1H-pyrazole
2-[(2E)-but-2-en-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
2-{4-[(3-methyl-1H-indol-2-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N1,N1-dimethyl-N3-[(3-phenylphenyl)methyl]piperidine-1,3-dicarboxamide
(1R,3s,6r,8S)-4-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(oxolane-3-carbonyl)piperidine
N-benzyl-N,1-dimethyl-5-({[3-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(3,3-diphenylpropyl)-6-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
4,6-dimethyl-2-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
N-[(2S)-4-methyl-1-{4-[4-methyl-2,5-dioxo-1-(thiophen-3-ylmethyl)imidazolidin-4-yl]piperidin-1-yl}-1-oxopentan-2-yl]acetamide
[(4aS,8aR)-1-(5-methyl-1,2-oxazole-4-carbonyl)-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(4-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
(3S,4R)-3-methoxy-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-amine
{3-[(4-fluorophenyl)methyl]-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl}methanol
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})(pyrazin-2-ylmethyl)amine
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-(furan-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[3-(2-methoxyphenoxy)propyl]-4,4-dimethylpyrrolidin-2-one
8-methoxy-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3,3-dimethyl-1-{[5-(thiophen-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
(5S,9aS,9bS)-5-(2,4-dimethoxyphenyl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(5-fluoropyrimidin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-cyclopropyl-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1,3-benzoxazole-6-carboxamide
N-[2-methyl-3-({methyl[(3-methylpyridin-4-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
4-[(3S,4S)-1-cyclobutanecarbonyl-4-hydroxypyrrolidin-3-yl]-1-phenylpiperazin-2-one