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2-(3-methoxypropyl)-8-(1-methyl-1H-indazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,5S)-1-benzyl-N-cyclohexyl-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[1'-(2-hydroxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-4-phenyl-N-(pyridin-3-ylmethyl)benzamide
(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)({[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl})amine
3-[(2,3-dihydroxypropyl)(methyl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
N-(2-fluoro-5-methylphenyl)-4-(3-methoxypropyl)piperazine-1-carboxamide
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
N-[(2,5-dimethoxyphenyl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
2-fluoro-N-[1-({[phenyl(pyridin-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(1S,6R)-3-[3-(piperazine-1-sulfonyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
3-hydroxy-N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)benzamide
14-[3-ethoxy-4-(propan-2-yloxy)phenyl]-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl 8-(2,2-diphenylethyl)-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}azepan-3-amine
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(1,2,5-thiadiazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[1-(2-phenylethyl)piperidin-3-yl]-4-(thiophen-2-yl)butanamide
ethyl 3-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]amino}propanoate
1-(2,3-dihydro-1H-inden-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)-2-methylpiperidine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
(2R,4S)-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-hydroxypiperidine-2-carboxylic acid
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-(piperidin-1-ylmethyl)benzamide
N-(2-methoxyethyl)-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-phenylpiperidin-3-amine
N-[1-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxypropanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(methylamino)pyridine-3-carboxamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(2-methylphenoxymethyl)piperidine
5-chloro-4-methyl-2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
7-(1-benzothiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,2-dimethylpropanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
1-[4-(benzyloxy)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-3-benzyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-4-{3-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-amino-7-[3-(1H-indol-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)acetamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
3-(phenoxymethyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide