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N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
7-(2-hydroxyethyl)-2-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(phenylamino)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-{2-oxo-2-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
6-(methoxymethyl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyridine-2-carboxamide
1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1,3-benzoxazole
N-[2-(2,4-difluorophenyl)-1-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
2-[3-(dimethylamino)propyl]-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(pyrrolidine-1-carbonyl)-5-[({[4-(trifluoromethoxy)phenyl]methyl}amino)methyl]phenyl]acetamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-3-ylmethyl)piperazine
(3aR,6aR)-2-methanesulfonyl-N-methyl-N-[(2-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-methylpiperazin-2-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
2-[(4-methoxyphenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]morpholine
4-cyano-N-[(3R,4S)-4-cyclopropyl-1-(6-methylpyridazin-3-yl)pyrrolidin-3-yl]oxane-4-carboxamide
2-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]-4-(trifluoromethyl)pyrimidine
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-1,2-oxazole-3-carboxamide
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2,6-dimethylquinoline-4-carboxamide
N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(morpholin-4-yl)benzamide
2-(2-fluoro-5-methoxyphenyl)-4-(3,3,3-trifluoropropyl)pyrimidine
1-[(2-fluorophenyl)methyl]-N-(2-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}benzoic acid
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(morpholin-4-yl)propan-1-one
N-[(3,4-difluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
N,2,3-trimethyl-N-(2-methylprop-2-en-1-yl)quinoxaline-6-carboxamide
3-{3-[2-(3-chlorophenyl)-1H-imidazol-1-yl]propyl}pyridine
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
(2S,4R)-1-benzyl-N-methyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(2-methoxyphenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-2-amine
2-ethyl-N-(1H-indol-4-ylmethyl)pyrimidine-5-carboxamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[2-(1H-indol-3-yl)ethyl]piperidin-4-amine
2-hydroxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
2-cyclopropyl-5-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(piperidin-1-yl)ethan-1-one
4-[(4-methoxyphenyl)methyl]-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one
N4,5-dimethyl-N4-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-2,4-diamine
(2S,4S)-4-amino-1-[4-(1H-imidazol-1-yl)butanoyl]pyrrolidine-2-carboxylic acid