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N-(1H-indol-5-ylmethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
5-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-(3-methylbutyl)imidazolidine-2,4-dione
N-{1-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
methyl 2-[2-(6-hydroxy-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)phenoxy]acetate
6-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-[(6-ethoxypyridin-3-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidin-4-ylmethyl)benzamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyrrolidin-3-yl)pyridin-2-amine
ethyl 5-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-ylmethyl}furan-2-carboxylate
(4aR,7aS)-1-(2-methylpropyl)-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(6-methylquinolin-5-yl)methyl]-4-(piperidin-1-yl)butanamide
3-ethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-4-carboxamide
2-[5-(1H-imidazol-2-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
4-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)pyridine
5-[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
2-amino-4-(furan-3-yl)-6-(1-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-ethyl-6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N-methylpyridine-3-carboxamide
5-(azepane-1-carbonyl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-[4-(benzyloxy)piperidin-1-yl]-2-ethoxyethan-1-one
1-(butan-2-yl)-N3-ethyl-4-oxo-N5-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-[(thiophen-3-ylmethyl)({[6-(trifluoromethyl)pyridin-3-yl]methyl})amino]butan-1-ol
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-1-carboxamide
3-(1,3-benzothiazol-2-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
(1S,4S)-2-(2-methyl-1,3-benzothiazol-5-yl)-5-(thiophen-3-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
8-[(4-fluoro-3-methylphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1H-indol-7-ylmethyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
4,4,4-trifluoro-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]butan-1-one
3-{[4-(dimethylamino)phenyl]methyl}-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[1-(7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclopropanecarboxamide
N-[3-(pyridin-4-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(2S,4S)-4-benzamido-N-ethyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-2-carboxamide
3-fluoro-N-[7-oxo-5-(4-propylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]benzamide
1-{[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]methyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-{3-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}propan-1-one
2-(4-chloro-2-methylphenoxy)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-[(4-methoxyphenyl)methyl]-1H-1,3-benzodiazole
3-{[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-cyclobutyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[2-(propan-2-yloxy)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]acetamide
2-[4-methyl-6-(4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-yl]phenol
ethyl 5-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
N-({1-[(2-chloro-5-fluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)furan-2-carboxamide
6-[2-(4-fluorophenoxy)ethyl]-2-(methylsulfanyl)pyrimidin-4-amine
1-[(3-fluorophenyl)methyl]-4-[(pyridin-4-ylmethyl)amino]pyrrolidin-2-one