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4,4,4-trifluoro-N-[(3R,4S)-1-(furan-2-ylmethyl)-4-propylpyrrolidin-3-yl]butanamide
N-(3-{5-methyl-4-[(2-oxo-2-phenylacetamido)methyl]-1,3-oxazol-2-yl}phenyl)-3-(pyridin-3-yl)propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-phenoxyphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-(2-methoxyacetyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
4-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
(4aR,7aS)-1-ethyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-chloro-5-methylbenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
N3-[2-(3-methoxyphenyl)ethyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-1-(6-ethoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
4-[4-(thiomorpholine-4-sulfonyl)benzoyl]morpholine
N-(4-chloro-2-fluorophenyl)-2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}acetamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(morpholin-4-yl)pyridine-3-carboxamide
{[3-(3-fluorophenyl)oxolan-3-yl]methyl}({[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
(3S,4S)-1-[2-(benzyloxy)ethyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-methyl-5-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-{3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
dimethyl({4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-oxazepan-6-yl}methyl)amine
(1R,5R)-3-methanesulfonyl-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
1-{2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-2-oxoethyl}pyrrolidin-2-one
ethyl 4-({3-[2-(methylcarbamoyl)ethyl]phenyl}carbamoyl)piperazine-1-carboxylate
4-(2-methyl-1H-imidazol-1-yl)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine-4-carboxylic acid
2-methoxy-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)pyridine-3-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-3-ylmethyl)amine
3-(2,3-dimethoxyphenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)pyrrolidine-1-carboxamide
1-{2-[methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]ethyl}cyclopentan-1-ol
N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-ethyl-1,2-oxazole-3-carboxamide
2-methoxy-N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-(1H-indazol-6-yl)-5-methylpiperazin-2-one
3-(2-chlorophenyl)-3-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
1-(4-methoxybenzoyl)-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
2-(3-{[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
N-(2-ethylphenyl)-3-{[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]amino}propanamide
1-cyclohexyl-4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
3-[2-(2,4-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
methyl (2S,4S)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(2,5-difluorophenyl)methyl]pyrrolidine-2-carboxylate
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
N-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-({4-[(3-phenoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
2,6-diamino-4-[2-(propylsulfanyl)pyrimidin-5-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[6-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide