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N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(1S,6R)-9-{[3-(2-hydroxyethoxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(carbamoylamino)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
6-[4-(dimethylamino)phenyl]-9H-purin-2-amine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
N-(2-methyl-1-{7-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)propanamide
1-[2-(2,3,4-trimethoxyphenyl)phenyl]piperazine
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
4-(1-acetylpiperidine-4-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]urea
3-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
(1R,5S)-8-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octane
1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
N-[(1-ethyl-1H-indazol-3-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
4-methyl-5-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
N,N-dimethyl-2-(4-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}morpholin-3-yl)acetamide
1-({5-[(3-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(1-phenylethyl)benzamide
8-(5-hydroxypyrazine-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
4-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}pyrimidin-2-amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(4-methoxyphenyl)-N-(oxolan-2-ylmethyl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
methyl 5-(quinoxaline-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-(4-chloro-2-methoxyphenoxymethyl)-N-(1-propylcyclopropyl)-1,2-oxazole-3-carboxamide
(2S,4S)-4-amino-1-[2-(2,2-dimethylpropanamido)-5-methylthiophene-3-carbonyl]-N-methylpyrrolidine-2-carboxamide
2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}propanamide
(1R,5S,6R)-3-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-(3-fluoro-4-methoxybenzoyl)-1-methylpiperidine
methyl 4-(5-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-(3-methylphenyl)-3-{1-[3-(2-oxopiperidin-1-yl)propanoyl]piperidin-4-yl}propanamide
5-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)-5-(thiophen-3-ylmethyl)pyrrolidin-2-one
1-[5-(2-chlorophenyl)furan-2-carbonyl]azetidine-2-carboxylic acid
5-cyano-6-(2,4-dimethoxyphenyl)-2-methylpyridine-3-carboxylic acid
1-[2-(2-fluoro-5-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
2-{[3-(propan-2-yloxy)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
{2-[(6-ethylpyrimidin-4-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)propylamine
1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-N,N-diethylpiperidine-4-carboxamide
5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-propylpyrimidine
1-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]piperidin-2-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]naphthalene-1-carboxamide
3-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-(adamantan-1-yl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
6-(2,3-dihydro-1-benzofuran-7-yl)-1H-[1,2,3]triazolo[4,5-b]pyridine
(1R,2S)-N1-butyl-N2-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexane-1,2-dicarboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine