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7-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(pyridin-2-ylmethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-amine
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
5-fluoro-1,3-dimethyl-2-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1H-indole
4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-1-[4-(1H-pyrazol-5-yl)phenyl]piperidine
(2S,4R)-4-amino-N-ethyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidine-2-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1,2-oxazinan-2-yl)propanamide
4-{7-fluoro-2-[2-(methylamino)pyrimidin-5-yl]quinoline-4-carbonyl}-1,3-dimethylpiperazin-2-one
4-(3-hydroxy-3-methylbutyl)-N-[3-(methylsulfanyl)propyl]benzamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-4-(morpholin-4-yl)-N-(oxolan-2-ylmethyl)benzamide
N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-benzyl-N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N6-(2-methoxyethyl)-N5-methyl-N5-(2-phenoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
methyl 5-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(3-chloro-5-fluorophenyl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
4-{[(3-hydroxy-3-phenylpropyl)(methyl)amino]methyl}-6,8-dimethyl-2H-chromen-2-one
2-[4-(4-benzylpiperazine-1-carbonyl)-5-(propan-2-yl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
1-(2-methylpropyl)-6-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]piperidine-3-carboxamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
9-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-(dimethylamino)-2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
7-[(3-methoxyphenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(furan-2-ylmethyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxamide
7-[3-(N-methylmethanesulfonamido)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
N-butyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
(3aR,7aS)-2-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-[(2-chlorophenyl)methyl]-5-[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
methyl 6-[(2,5-dimethylphenyl)methyl]-2-[(propan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2R,3R)-3-[4-(2,2-dimethoxyethyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-amino-2-{4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-1-yl}pyrimidine-5-carbonitrile
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylquinoline-4-carboxamide
(2R,6R)-4-(5-hydroxypyrazine-2-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(naphthalen-1-yl)acetamide
ethyl 4-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-3-yl}piperazine-1-carboxylate
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N,N-dimethyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]quinoxaline-6-carboxamide
2-acetyl-8-(quinolin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2R,3S,6R)-3-(2,3-difluorophenyl)-N,N-diethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
1-{1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-yl}azepane
1-[(3-chlorophenyl)methyl]-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
1-{3-[4-(1,2,3,6-tetrahydropyridin-1-yl)piperidin-1-yl]phenyl}imidazolidin-2-one