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2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-N-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
6-ethyl-2-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
[(2S,6S)-11-methoxy-4-(pent-2-yn-1-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
6-chloro-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
(4aR,7aS)-1-benzyl-4-[(3-hydroxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclobutanecarboxamide
3-[4-(5-cyanopyridin-2-yl)piperazine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
1-cyclobutyl-5-methyl-5-phenylpiperidin-2-one
2-[3-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-1-yl]acetamide
1-[(4aS,8aS)-7-cyclohexyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-2-(1,1-dioxo-1λ6-thian-4-yl)acetamide
ethyl 2-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-2-yl)acetate
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)benzamide
6-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxylate
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-(trifluoromethoxy)benzene-1-sulfonamide
3-(4-chlorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
methyl 1-benzyl-3-(oxolane-2-amido)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,3S,5S)-8-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
4-(2,2-difluoroethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(diethylamino)-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1-methyl-1H-imidazole-5-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(3-methoxypropyl)-8-[(3-methylthiophen-2-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aR)-1-(2-aminoethyl)-6-(2-phenylethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-({5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-{3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}piperidin-2-one
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-2-ol
3-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[3-(2-fluorophenyl)propyl]piperazin-1-yl}pyrimidine
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
9-(propane-1-sulfonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-ethylpiperidine
1-(cyclopropylmethyl)-4-(6-methylpyridazin-3-yl)-2-(propan-2-yl)-1,4-diazepane
(5-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2-ethoxyphenyl)methanol
2-cyclohexyl-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1,3-benzoxazole-6-carboxamide
[(2-phenoxypyridin-3-yl)methyl][(1-phenyl-1H-pyrazol-4-yl)methyl]amine
(3-{2-[1-(4-ethenylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(4-methoxy-3-methylphenyl)methyl]piperidine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(1H-1,3-benzodiazol-1-yl)propan-1-one
2-[4-(pyridin-4-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-[(dimethylamino)methyl]-1-(6-ethyl-2-methylquinoline-4-carbonyl)azepan-4-ol