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1-(2-aminopyrimidin-4-yl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
3-methyl-1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]butan-1-ol
5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-[(2-fluorophenyl)methyl]-5-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{4-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}ethan-1-one
2-[4-(2-methyl-5-propylpyrimidin-4-yl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine-2,6-dione
(3S,4S)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-2-yl)acetamide
7-[2-(propan-2-yloxy)phenyl]-1,2,3,4-tetrahydroisoquinoline
2-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-1-propyl-1H-imidazole
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N,N-dimethyl-4-oxobutanamide
3-[(4aR,7aS)-4-[(3-methoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-({[3-(dimethylamino)-2,2-dimethylpropyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-(2-chlorophenyl)-3-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
2-{[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]methyl}-2,8-diazaspiro[4.5]decane
(2S,4S,5R)-4-[(furan-3-ylmethyl)(methyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
2-cyclopropyl-5-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyrimidine
5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-hydroxypropan-1-one
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methanesulfonylethyl)piperazine
3-(3-chlorobenzoyl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
4-(azepan-1-yl)-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-cyclopropyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-methyl-1H-pyrazole-4-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
4-(4-benzyl-1H-pyrazol-5-yl)-1-(3-methylpiperidine-3-carbonyl)piperidine
7-(cyclopropylmethyl)-2-(1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-(3,3-diphenylpiperidin-1-yl)-2-(morpholin-2-yl)ethan-1-one
5-({4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
5-(3,4-difluorophenoxymethyl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1,2-oxazole-3-carboxamide
8-[3-(2-oxopiperidin-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N-methylthiophene-2-carboxamide
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 1-{1-[4-(2-phenoxyacetamido)phenyl]piperidin-4-yl}piperidine-3-carboxylate
8-cyclobutyl-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenyl]acetamide
1-(furan-3-ylmethyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-6-ol
N-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(furan-2-ylmethyl)-N-[(2-hydroxyphenyl)methyl]-N-methylpiperidine-3-carboxamide
1-[(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
4-(4-methylpiperazin-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
(3S,4S)-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclopentyl-N3-(2-methylpropyl)-N5-[2-(methylsulfanyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(1,4-dioxane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-2-methyl-6-(trifluoromethyl)pyridine