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6-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyrimidin-2-amine
2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-5-methoxyphenol
3-butanamido-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]benzamide
1-[(5-chloro-2-hydroxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperazine
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
methyl 5-(4-{[4-(1,3-benzoxazol-2-yl)phenyl]carbamoyl}piperidin-1-yl)-5-oxopentanoate
6-(4-fluorophenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[2-(dimethylamino)ethyl]-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aS)-1-(3-ethoxypropyl)-6-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-(pyrimidin-2-yl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
methyl 5-{[(2,3-dimethoxyphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-3-(piperidin-1-ylmethyl)piperidine
8-(2,5-dimethylfuran-3-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-fluoro-N-[2-(2-methoxyphenyl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-{[7-(2-chloro-4-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
2-(2-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
3-(5-chloro-2-methoxybenzoyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(3,4-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-methylthian-4-amine
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N'-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]-N-(2,5-dimethylphenyl)propanediamide
N-[3-(1H-indol-2-yl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
N-methyl-5-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}-1,2,4-oxadiazole-3-carboxamide
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methylpyridine
N-cyclopropyl-3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-{[({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
1-(2,6-dimethylphenyl)-3-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]urea
4-{[1-(thiophene-3-carbonyl)piperidin-2-yl]methyl}morpholine
3,4,5-trimethoxy-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]benzamide
1-ethyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(pyridin-3-yloxy)propyl]acetamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(thiophene-2-carbonyl)piperazine
1-[2-(4-fluorophenyl)ethyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
1-[(3-chlorophenyl)methyl]-4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
5-(1H-indol-1-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
1-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
6-(cyclopropylmethoxy)-4-(2,3-dihydro-1H-inden-2-yl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
N3-cycloheptyl-1-cyclopropyl-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-methylquinolin-2-yl)piperidin-3-yl]propan-1-ol
(1S,9R)-11-{[3-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(4-{[2-(ethylsulfanyl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one