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5-fluoro-2-[3-({[1-(3-methoxyphenyl)ethyl](methyl)amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
(3R,5S)-5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-3-ol
(3S,4S)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-({[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
5-({[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
N-{[1-(1,3-dihydroxypropan-2-yl)piperidin-3-yl]methyl}-2-hydroxy-5-methylbenzamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(3-phenylpropyl)amine
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-N'-(2-methylphenyl)propanediamide
6-(pyrrolidin-1-ylmethyl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-oxazepan-6-ol
9-{[4-(2-hydroxyethoxy)phenyl]methyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-ethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
(1S,5R)-6-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
({3-[2-(2-ethylpyrimidin-4-yl)-1H-imidazol-1-yl]phenyl}sulfamoyl)dimethylamine
2-(diethylamino)-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
2-(3-phenylpropyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
3-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-(2-methyl-5-sulfamoylphenyl)urea
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-(2,6-dimethylpyridin-4-yl)-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
4-(1,3-thiazol-2-ylmethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
dimethyl[2-({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
(2R,6R)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidine-3-carboxylic acid
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
4-methyl-2-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-[(isoquinolin-5-yloxy)methyl]-N-(oxolan-2-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
6-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
1-[2-(benzyloxy)phenyl]-3-[3-(4-hydroxypiperidin-1-yl)propyl]urea
2-{[(2-methylphenyl)methyl]sulfanyl}-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
N-tert-butyl-1-cyclohexyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
naphthalen-1-yl (7R,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(2R,3S,6R)-5-(1H-indole-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
N-(propan-2-yl)-5-(thiomorpholine-4-carbonyl)pyrimidin-2-amine
4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
3-butyl-1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-3-(3-ethylphenoxy)azetidine
N,2-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5-(propan-2-yl)furan-3-carboxamide
N-(1H-indazol-7-yl)-4-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carboxamide
4-[4-ethyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
3-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
dimethyl({[(3S,4R)-1-(6-methyl-2-propylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
2-(6-methoxynaphthalen-2-yl)-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]morpholine
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[2-(4-methyl-1H-imidazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
10-methoxy-5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[3-(morpholin-4-yl)azetidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,3-benzodiazole-6-carboxylic acid