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1-[(4-fluorophenyl)methyl]-N-[1-(naphthalen-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-2-amine
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(2-phenylpropyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-5-(methoxymethyl)thiophene-2-carboxamide
3-(2-hydroxyphenyl)-N-(2-phenylethyl)-N-propyl-1H-pyrazole-5-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-{[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,5-dimethyl-1H-pyrazole
1-methyl-N-[3-(pyridin-4-yl)propyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4S)-4-cyclopropyl-1-[(methylcarbamoyl)methyl]pyrrolidin-3-yl]-3-(3-methoxyphenyl)propanamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(pyridin-4-yl)propyl]propanamide
5-[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]-1H-imidazole-4-carboxylic acid
6-(2-chlorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(3,4,5-trimethoxyphenyl)acetamide
1-(1,3-benzothiazol-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-3,4-dimethoxybenzamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
2-(2-oxopyrrolidin-1-yl)-N-[3-(3-phenylpropanamido)phenyl]propanamide
6-(4-methylphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethylurea
3-methyl-7-{[4-(pyridin-2-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(2-methoxyphenyl)methyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanamide
N-cycloheptyl-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-yl)-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-({[(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
2-cyclopropyl-1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methylpyrrolidine-2-carboxamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
(1S,5R)-6-(2,4-difluorobenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
5-(2-methoxyacetamido)-1-methyl-N-[(1-phenylcyclopentyl)methyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-7-methylquinolin-3-yl)methanol
1'-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
6-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
3-(2,4-dimethoxyphenyl)-2-methyl-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
3-({[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amino}methyl)-N,N-dimethylpyridin-2-amine
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
5-[1-(adamantane-1-carbonyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
4-hydroxy-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(3R,5R)-1-(4-fluoro-3-methylbenzoyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol