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1-(2-ethoxyethyl)-5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{[(cyclopropylmethyl)(propyl)amino]methyl}-4-(3,6-dimethylpyrazin-2-yl)phenol
1-(4-chloro-1H-pyrrole-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
N-[2-(2-chlorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
(3S)-1-(2-methoxypyridine-4-carbonyl)-N,N-dimethylazepan-3-amine
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
6-[4-(5-methyl-2-phenylfuran-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
methyl[(4-{2-[1-(1-methylpiperidine-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
1-ethyl-6-oxo-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(4-methylphenyl)propanamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
(3R,4R)-1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-cyclobutyl-4-methylpyrrolidin-3-ol
4-{5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}benzonitrile
N-[3-(dimethylamino)-1-phenylpropyl]pyrimidin-2-amine
ethyl 2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]acetate
2-(2-methyl-1-benzofuran-7-carbonyl)-1,2,3,4-tetrahydroisoquinoline
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-ol
N-(1-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
2-(4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-1-methylpiperazin-2-yl)ethan-1-ol
3-(2-methoxyethyl)-1-[4-(thiophen-2-yl)butanoyl]piperidine-3-carboxylic acid
(3R,4S)-4-cyclopropyl-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]pyrrolidin-3-amine
2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]-N-(oxolan-2-ylmethyl)acetamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[(3R,4R)-1-(2,3-dimethoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}methyl)furan-2-carboxamide
6-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
3-methyl-7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[2-({[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-5-fluorobenzonitrile
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(2-methoxyethyl)-7-(pyridine-3-amido)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
{3-[2-(furan-2-yl)-1H-imidazol-1-yl]-3-phenylpropyl}dimethylamine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-methyl-8-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-5-tert-butyl-1H-pyrazole
methyl 3-(pent-4-enamidomethyl)-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N2-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N4-ethylpyrimidine-2,4-diamine
3-[(3R,4S)-1-(3-hydroxy-4-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N4-[(2-chlorophenyl)methyl]-N4-methyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl]propanoate
(3R,4S)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-propylpyrrolidin-3-amine
1-(4-methoxyphenyl)-4-(piperidin-3-yl)piperazine
N,N-dimethyl-4-oxo-4-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)butanamide
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-[2-(cyclohex-1-en-1-yl)ethyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one