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6-(2,5-dimethylphenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
(2R,3R)-3-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]propanamide
N-(1-{6-[(2-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-3-methyl-1-oxobutan-2-yl)acetamide
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxypyridin-4-ol
ethyl 4-[5-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-7-carbonyl]piperazine-1-carboxylate
4-(propylsulfamoyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
N-[(2R,3R)-1'-[3-(4-methylphenyl)propanoyl]-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-(2-methoxy-4-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(1-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
9-(cyclopropylmethyl)-1-methyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-({1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperidin-4-yl}oxy)benzoic acid
6-(1H-indol-4-yl)-4-(4-methylpiperazin-1-yl)quinazoline
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-{1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-4-yl}-3-methylbutan-1-ol
6-cyano-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}pyridine-3-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
(3S,4R)-1-(1H-indol-4-ylmethyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-2,2-diphenyl-N-(pyridin-3-ylmethyl)acetamide
N-(2-methoxyethyl)-1-methyl-5-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrrole-2-carboxamide
(7S,9aR)-N-cyclohexyl-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[(5-oxopyrrolidin-2-yl)methyl]-1-(3-phenylpropyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-{1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[2-(2-phenylquinazolin-4-yl)ethyl]-1λ6-thiolane-1,1-dione
7-methanesulfonyl-2-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidin-1-yl}-2-phenoxyethan-1-one
3-({7-acetyl-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)-N-(4-fluorophenyl)propanamide
3-(2-methoxyethyl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine-3-carboxylic acid
N-cyclohexyl-2-[4-(pyridin-4-yl)piperidin-1-yl]butanamide
2-(2,5-dimethoxyphenyl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-cyano-N-cycloheptyl-N-ethylbenzamide
(1S,5R)-3-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
1-[3-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
2-[benzyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
3-(5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-N-[(4-methylphenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(pyridin-3-yl)piperazine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[4-(hydroxymethyl)phenyl]methyl}-5-methylpiperidin-2-one
N-[(4-fluorophenyl)methyl]-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
4-(4-{1-[2-(ethylsulfanyl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-3-methyl-1H-1,2,4-triazole
N-[2-oxo-4-(quinolin-4-yl)-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
N-(2-{1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinolin-6-yl)acetamide