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3-(cyclopropylmethyl)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]piperidine-3-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-phenyl-1,2,4-oxadiazol-5-amine
N-ethyl-N-(2-methylprop-2-en-1-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
6-(4-fluorophenyl)-N-{[1-(methoxymethyl)cyclopropyl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4S)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
(2,3-dihydro-1-benzofuran-5-ylmethyl)(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-[1-(benzenesulfonyl)piperidin-4-yl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
N-[3-(4-{[(1S)-1-carbamoyl-2-phenylethyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
N-ethyl-2-oxo-2-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-ethyl-N-[2-(quinolin-8-yloxy)ethyl]pyrimidine-5-carboxamide
N,7,8-trimethyl-N-(oxan-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-[2-(2-methoxyethoxy)acetyl]piperazin-2-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(pyridin-3-yl)acetamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidine-2-carboxamide
N-[4-(4-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
(1R,5S,8R)-8-methoxy-3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-azabicyclo[3.2.1]octane
1-{4-[3-cyclopropyl-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}-3-methylbutan-1-one
2-(4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
8-(ethanesulfonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-(4-phenyl-1,3-thiazol-2-yl)-5-({[1-(thiophen-2-yl)propyl]amino}methyl)-1H-pyrazole-4-carboxylate
(4aS,8aR)-6-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
8-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
1-(3-phenylpropyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(1-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
3-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-indol-2-one
N-[2-(diethylamino)ethyl]-N-methyl-2-(4-methylpiperazin-1-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
1-[2-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-(5-fluoro-2-methylphenyl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
3-{[4-(furan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-7-methylquinolin-2-ol
ethyl 2-(4-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}morpholin-3-yl)acetate
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
3-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
5-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
4-(2-chloro-4-fluorophenyl)-2-methylquinazoline
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
3-cyclohexyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2,6-difluorophenyl)-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
4-[(2R)-2-hydroxypropanoyl]-1-(4-methylphenyl)piperazin-2-one
2-[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
5-[(5-chlorofuran-2-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(furan-2-ylmethyl)-1-methylurea
6-methoxy-N,3-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
2-[1-(2-phenylethyl)-4-[4-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]ethan-1-ol
4-methyl-N-[3-(methylsulfamoyl)phenyl]-3-phenylpiperazine-1-carboxamide
N-{4-[4-({[2-(dimethylamino)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-5-(methoxymethyl)furan-2-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
4-(4-chlorophenoxy)-N-(2-oxoazepan-3-yl)piperidine-4-carboxamide