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2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]morpholin-3-yl}-1-(thiomorpholin-4-yl)ethan-1-one
N3-[(2-chlorophenyl)methyl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidin-3-amine
(1R,3S)-7-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
6-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
3-{methyl[4-(pyridin-3-yl)pyrimidin-2-yl]amino}propan-1-ol
4-(5-methylpyrimidin-2-yl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane
2-(adamantan-1-yl)-5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
5-methyl-1-(2-methylphenyl)-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
(3aS,6aS)-2-(2-methoxyethyl)-5-[(2-methoxynaphthalen-1-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3-fluorophenyl)methyl]-5-(4-methoxypiperidine-1-carbonyl)piperidin-2-one
1-[(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-cyclopentyl-1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
2-(4-hydroxyphenyl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidin-2-amine
1-(morpholine-4-carbonyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
2-methyl-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
(2S,4S)-4-amino-1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
7-(2-methylphenyl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(1-benzothiophen-2-yl)-N-[2-(diethylamino)ethyl]-N-methyl-2-(morpholin-4-yl)pyridine-3-carboxamide
1-{3-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
N-[4-(2-fluorophenoxy)phenyl]-1-(2-hydroxyacetyl)piperidine-4-carboxamide
ethyl 4-{7-[1-(2-fluorophenyl)-4-hydroxypiperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidine-1-carboxylate
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[({[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
1-[2-(2-fluorophenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
1-cyclohexyl-N3-[(4-methoxyphenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-cyclohexyl-4-[(2E)-4-methylpent-2-en-1-yl]piperazin-2-yl}ethan-1-ol
4-(3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-methylpyrimidine
4-{1-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}benzene-1-sulfonamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
N,2,6,8-tetramethyl-N-[1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
5-{[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methanesulfonamido-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-[(3-methoxyphenyl)sulfanyl]-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]acetamide
2-(2,2-dimethyloxan-4-yl)-1-[(5-fluoro-2-methylphenyl)methyl]-1H-imidazole
(3S,4R)-4-(2-methoxyphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxylic acid
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-(oxolan-2-ylmethyl)-1-(thiophen-3-ylmethyl)urea
cyclopentyl 4-[(2S)-2-amino-3-methoxypropanamido]benzoate
[(3-fluoro-2-methylphenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
7-(1,3-benzothiazol-2-yl)-4-[(2,6-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}pyridine-4-carboxylic acid
6-{[(2-methylphenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
9-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one