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4-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-3-(3-fluorophenyl)piperazin-2-one
3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[4-(4-{[2-hydroxy-3-(3-methoxyphenoxy)propyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
(1S,5R)-3-benzyl-6-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(pyridin-3-yloxy)acetamide
8-(5-methylpyrazine-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1H-indol-5-yl)-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
({5-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]thiophen-3-yl}methyl)dimethylamine
3-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
(3S)-1-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]acetamide
2-(1,2-benzoxazol-3-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}acetamide
(1R,2S,6R,7S)-4-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
1'-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(2,5-dimethylphenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-{1'-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
N-({7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
N-tert-butyl-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-(1H-imidazol-2-yl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol
1-(cyclohexylmethyl)-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
(3S,4S)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-[(3-fluorophenyl)methyl]-4-(1-methyl-1H-imidazole-5-carbonyl)piperazine
4-oxo-6-[(1E)-pent-1-en-1-yl]-1,4-dihydroquinoline-3-carboxylic acid
2,6-difluoro-N-({7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-(4-{1-[3-(3-methoxyphenyl)phenyl]piperidin-4-yl}morpholin-2-yl)ethan-1-ol
N-[(4-fluorophenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-(4-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}phenyl)acetamide
2-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]pyridine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
2-fluoro-6-methoxy-N-(3-phenylprop-2-yn-1-yl)-N-propylbenzamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
7-fluoro-N,2-dimethyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)quinoline-4-carboxamide
3-{4-[(3-methylquinoxalin-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)acetamide
3-methyl-1-{1-[6-(1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
2-[(3-fluorophenyl)methyl]-4-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
6-methyl-2-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
3-(2,6-dimethoxypyridine-3-carbonyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3aR,6aR)-2-(ethanesulfonyl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-{1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-methoxy-5-oxo-6-[2-(2-oxoimidazolidin-1-yl)ethyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
3-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3,4-dihydropteridin-4-one
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-phenyl-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine