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1-cyclopropanecarbonyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
(1H-imidazol-2-ylmethyl)(methyl){[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
2-(pyridin-4-ylsulfanyl)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
3-benzyl-1-(3-methoxypropyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-benzyl-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperazin-2-one
1-{[(3R,4R)-4-(hydroxymethyl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(2,4-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
6-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
5-[2-(aminomethyl)-4-fluorophenyl]thiophene-2-carboxamide
2-[(2,4-difluorophenyl)methyl]-8-methyl-2,8-diazaspiro[4.5]decane
1-[1-(5-fluoro-2-methylbenzoyl)piperidin-4-yl]-2-phenylethan-1-ol
N-tert-butyl-3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propanamide
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-5-methoxyphenol
7-(2,6-dimethoxyphenyl)-9-methoxy-4-[(1-methyl-1H-indol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2E)-3-(3,4-dimethoxyphenyl)-1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}prop-2-en-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
2-({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N,N-dimethylpropanamide
5-ethyl-3-(1-hydroxyhexan-2-yl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-(quinolin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(5-{[3-(2-fluorophenoxymethyl)piperidin-1-yl]methyl}furan-2-yl)methanol
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methylacetamide
(2R,3R,6R)-5-(3-fluoropropyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)-1,3-benzothiazole
2-butyl-N-(1H-indazol-5-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
2,5-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]methyl}benzoic acid
7-(2-aminopyridine-4-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-hydroxy-1-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperidine-4-carboxylic acid
5-(hydroxymethyl)-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}furan-2-carboxamide
N-[2-(2-methyl-1-benzofuran-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
methyl 1-benzyl-5-[(3-hydroxybutyl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4R)-4-amino-1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methylpyrrolidine-2-carboxamide
2-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-N-(pyridin-2-ylmethyl)aniline
1-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)propanamide
N-[4-(4-{[(2,4-dimethylphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
N-cyclooctyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(1,2-oxazol-3-ylmethyl)piperidin-3-amine
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzoyl]piperidin-3-ol
[(2,2-dimethyloxan-4-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
[3-(cyclopropylmethyl)-1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]methanol
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(1-methyl-1H-indole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2,6-dimethylphenoxymethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-5-(1H-indole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3,4-difluorophenyl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[2-(methylsulfanyl)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one