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N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-methoxypiperidine-1-carboxamide
2-(diethylamino)-1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}ethan-1-one
3-{2-[methyl(quinoxalin-2-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-fluoro-4-hydroxy-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}quinoline-3-carboxamide
5-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}benzamide
{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-[(2-fluorophenyl)methyl]-1-(2-hydroxyethyl)-N-(pentan-3-yl)-1H-1,3-benzodiazole-5-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)propylamine
3,4,7-trimethyl-2-(3-phenoxyazetidine-1-carbonyl)-1H-indole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-methyl-1,3-thiazole-4-carboxamide
N'-[2-(dimethylamino)ethyl]-N'-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-N,N-dimethylbutanediamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-({5-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
5-chloro-N-(1-methylpiperidin-4-yl)-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-[4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
1-(4-acetylpiperazin-1-yl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-{2-[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4'-butyl-1-(3,3-dimethylbutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-(2-fluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
N-(3-methoxypropyl)-6-(2-methyl-4-phenylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[2-(4-chlorophenyl)-2-hydroxyacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-(2,4-difluorophenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
1-{2-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
4-(4-chlorophenyl)-N-[(2,5-difluorophenyl)methyl]butanamide
5-fluoro-2-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
8-(1-benzofuran-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-1-(2-methylpropyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-(3-carboxy-5,6-dimethylpyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
N-(2-fluoro-5-{[(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)carbamoyl]amino}phenyl)acetamide
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-(pyridin-3-yl)morpholine
methyl (2S)-3-methyl-2-{[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
1-(4-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
2-acetyl-8-[2-(3-methoxyphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(4-chloro-2-fluorophenyl)-1-ethyl-3-methyl-1H-1,2,4-triazole
3-(3-benzylpyrrolidine-1-carbonyl)-5-propyl-1,2-oxazole
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide