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4-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine-4-carbonyl}morpholine
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(4-methyl-3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-cyclooctyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(2S,4R)-N-[2-(3-chlorophenyl)ethyl]-1-[(4-fluorophenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(2-methylpyridin-4-yl)methyl]quinoline-4-carboxamide
3-{1-[(3-chloropyridin-4-yl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
N1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-N2-methylpyrrolidine-1,2-dicarboxamide
(1R,5R)-6-[2-(2-chloro-6-fluorophenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(3S,4R)-3-acetamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
6-[(2-fluorophenyl)methoxy]-4-(2-hydroxy-2-methylpropanoyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
4-(1-benzofuran-2-carbonyl)-1-cyclohexyl-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-({3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1λ6-thiolane-1,1-dione
1-[(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
(1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
1-(4-chlorophenyl)-3-{[1-(hydroxymethyl)cyclobutyl]methyl}urea
1-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)-4-methylpiperidine-4-carbonitrile
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-ethoxyfuran-2-carbonyl)pyrrolidin-3-yl]methanol
(4aS,7aR)-1-(2-butoxyacetyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-(2-methoxyethoxy)piperidine
(3S,4S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
(1R,6S)-3-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{imidazo[1,2-a]pyridin-2-ylmethyl}acetamide
1-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
(1R,5S)-3-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(morpholin-4-yl)benzamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-amino-6-(2-methylphenyl)-4-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
ethyl 1-(2,3-dimethylphenyl)-5-{[(2-acetamidoethyl)amino]methyl}-1H-pyrazole-4-carboxylate
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
7-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
6-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazin-2-amine
5-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-cyclopentyl-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}quinoline-2-carboxamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N,2,6-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}quinoline-4-carboxamide
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)(pyrazin-2-ylmethyl)amine
[4-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-(dimethylamino)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
5-(4-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}phenoxy)-1H-1,2,3,4-tetrazole
5-methyl-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-2-(3-methylphenyl)-1,3-oxazole
2-{1-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]propanamide
2-(methoxymethyl)-N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid